Journal Articles
2018
Induction of cell killing and autophagy by amphiphilic pyrrolidine derivatives on human pancreatic cancer cells
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. 2018.
DOI : 10.1016/j.ejmech.2018.02.086.
2016
Organocatalysis: Fundamentals and Comparisons to Metal and Enzyme Catalysis
Catalysts. 2016.
DOI : 10.3390/catal6090128.
1,2,3-Triazoles as inhibitors of indoleamine 2,3-dioxygenase 2 (IDO2)
Bioorganic & Medicinal Chemistry Letters. 2016.
DOI : 10.1016/j.bmcl.2016.07.031.
Synthesis and Applications of Silyl 2-Methylprop-2-ene-1-sulfinates in Preparative Silylation and GC-Derivatization Reactions of Polyols and Carbohydrates
Chemistry-A European Journal. 2016.
DOI : 10.1002/chem.201504380.
2015
Challenges in the Discovery of Indoleamine 2,3-Dioxygenase 1 (IDO1) Inhibitors
Journal Of Medicinal Chemistry. 2015.
DOI : 10.1021/acs.jmedchem.5b00326.
2014
The anti-lymphoma activity of APO866, an inhibitor of nicotinamide adenine dinucleotide biosynthesis, is potentialized when used in combination with anti-CD20 antibody
Leukemia & Lymphoma. 2014.
DOI : 10.3109/10428194.2013.869325.
Detailed analysis and follow-up studies of a high-throughput screening for indoleamine 2,3-dioxygenase 1 (IDO1) inhibitors
European Journal Of Medicinal Chemistry. 2014.
DOI : 10.1016/j.ejmech.2014.06.078.
A critical role of autophagy in antileukemia/lymphoma effects of APO866, an inhibitor of NAD biosynthesis
Autophagy. 2014.
DOI : 10.4161/auto.27722.
Synthesis Of Pyrrolidine 3,4-Diol Derivatives With Anticancer Activity On Pancreatic Tumor Cells
Heterocycles. 2014.
DOI : 10.3987/Com-13-S(S)111.
Amides in One Pot from Carboxylic Acids and Amines via Sulfinylamides
Organic Letters. 2014.
DOI : 10.1021/ol403508j.
2013
Amide Formation in One Pot from Carboxylic Acids and Amines via Carboxyl and Sulfinyl Mixed Anhydrides
Organic Letters. 2013.
DOI : 10.1021/ol401053y.
2012
A C-Linked Disaccharide Analogue of Thomsen-Friedenreich Epitope Induces a Strong Immune Response in Mice
Chemistry-A European Journal. 2012.
DOI : 10.1002/chem.201200364.
Synthesis of branched seven-membered 1-N-iminosugars and their evaluation as glycosidase inhibitors
Carbohydrate Research. 2012.
DOI : 10.1016/j.carres.2011.10.039.
Rational Design of 4-Aryl-1,2,3-Triazoles for Indoleamine 2,3-Dioxygenase 1 Inhibition
Journal Of Medicinal Chemistry. 2012.
DOI : 10.1021/jm300260v.
Synthesis of 2-(1-aminocyclopropyl)pyrrolidine-3,4-diol derivatives applying titanium-mediated reaction conditions
Tetrahedron. 2012.
DOI : 10.1016/j.tet.2011.12.024.
Synthesis of a C-Iminoribofuranoside Analog of the Nicotinamide Phosphoribosyltransferase (NAMPT) Inhibitor FK866
Helvetica Chimica Acta. 2012.
DOI : 10.1002/hlca.201100415.
Chemical strategies for controlling protein folding and elucidating the molecular mechanisms of amyloid formation and toxicity
Journal of molecular biology. 2012.
DOI : 10.1016/j.jmb.2012.01.051.
2011
Anti-cancer activity of 5-O-alkyl 1,4-imino-1,4-dideoxyribitols
Bioorganic & Medicinal Chemistry. 2011.
DOI : 10.1016/j.bmc.2011.07.053.
The norbornene mystery revealed
Chemical Communications. 2011.
DOI : 10.1039/c0cc00601g.
Total Asymmetric Syntheses of beta-Hydroxy-delta-lactones via Umpolung with Sulfur Dioxide
Journal Of Organic Chemistry. 2011.
DOI : 10.1021/jo102035d.
Glycochemistry Today
Chimia. 2011.
Concise Synthesis of Complicated Polypropionates through One-Pot Dissymmetrical Two-Directional Chain Elongation
Chemistry-A European Journal. 2011.
DOI : 10.1002/chem.201003264.
Efficient Asymmetric Synthesis of Long-Chain Polyketides Containing up to Ten Contiguous Stereogenic Centres by Double Chain Elongation
European Journal Of Organic Chemistry. 2011.
DOI : 10.1002/ejoc.201100196.
2010
Structural Insights into the Specificity of Xyn10B from Paenibacillus barcinonensis and Its Improved Stability by Forced Protein Evolution
Journal Of Biological Chemistry. 2010.
DOI : 10.1074/jbc.M109.064394.
Rational Design of Indoleamine 2,3-Dioxygenase Inhibitors
Journal Of Medicinal Chemistry. 2010.
DOI : 10.1021/jm9014718.
Novel 2-[(benzylamino)methyl]pyrrolidine-3,4-diol derivatives as alpha-mannosidase inhibitors and with antitumor activities against hematological and solid malignancies
Bioorganic & Medicinal Chemistry. 2010.
DOI : 10.1016/j.bmc.2010.03.009.
Synthesis and glycosidase inhibitory activity of 1-amino-3,6-anhydro-1-deoxy-D-sorbitol derivatives
Bioorganic Chemistry. 2010.
DOI : 10.1016/j.bioorg.2009.12.002.
BCl3-Mediated Ene Reaction of Sulfur Dioxide and Unfunctionalized Alkenes
Chemistry-A European Journal. 2010.
DOI : 10.1002/chem.201000164.
Synthesis of new oxathiazinane dioxides and their in vitro cancer cell growth inhibitory activity
Bioorganic & Medicinal Chemistry Letters. 2010.
DOI : 10.1016/j.bmcl.2009.09.019.
The Catalyzed Desulfinylative Allylation of Carbonyl Compounds with Alk-2-enesulfonyl Chlorides and Silyl Alk-2-enesulfinates
Chemistry-A European Journal. 2010.
DOI : 10.1002/chem.201000705.
The regioselectivity of the addition of benzeneselenyl chloride to 7-azanorborn-5-ene-2-yl derivatives is controlled by the 2-substituent: new entry into 3-and 4-hydroxy-5-substituted prolines
Tetrahedron. 2010.
DOI : 10.1016/j.tet.2010.06.090.
Stereoselective syntheses of polyhydroxylated azepane derivatives from sugar-based epoxyamides. Part 1: synthesis from D-mannose
Tetrahedron-Asymmetry. 2010.
DOI : 10.1016/j.tetasy.2010.06.035.
Synthesis, Biological Evaluation and Docking Studies of Casuarine Analogues: Effects of Structural Modifications at Ring B on Inhibitory Activity Towards Glucoamylase
European Journal Of Organic Chemistry. 2010.
DOI : 10.1002/ejoc.201000632.
Total Synthesis and Determination of the Absolute Configuration of (-)-Dolabriferol
Angewandte Chemie-International Edition. 2010.
DOI : 10.1002/anie.201003735.
Short Diastereoselective Synthesis of the C1-C13 (AB Spiroacetal) and C17-C28 Fragments (CD Spiroacetal) of Spongistatin 1 and 2 through Double Chain-Elongation Reactions
Chemistry-A European Journal. 2010.
DOI : 10.1002/chem.201002204.
Synthetic studies toward the CD spiroketal of spongistatins
European Journal of Organic Chemistry. 2010.
DOI : 10.1002/ejoc.200901285.
2009
Synthesis of Optically Active 5-Alkoxy-6-methylcyclohex-2-en-1-ones and 4-Alkoxy-5-methylcyclopent-1-enyl Benzoate
Journal Of Organic Chemistry. 2009.
DOI : 10.1021/jo801981c.
Synthesis of novel pyrrolidine 3,4-diol derivatives as inhibitors of alpha-L-fucosidases
Organic & Biomolecular Chemistry. 2009.
DOI : 10.1039/b819867e.
Umpolung with Sulfur Dioxide: Carbon-Carbon Cross-Coupling of Electron-Rich 1,3-Dienes and Alkenes; Application to the Enantioselective Synthesis of Long-Chain Polyketide Fragments
Synthesis-Stuttgart. 2009.
DOI : 10.1055/s-0028-1088011.
Design and synthesis of acetamido tri- and tetra-hydroxyazepanes: Potent and selective beta-N-acetylhexosaminidase inhibitors
Bioorganic & Medicinal Chemistry. 2009.
DOI : 10.1016/j.bmc.2009.06.022.
The spirocyclopropyl moiety as a methyl surrogate in the structure of L-fucosidase and L-rhamnosidase inhibitors
Bioorganic & Medicinal Chemistry. 2009.
DOI : 10.1016/j.bmc.2009.10.010.
Synthesis of (E,Z)-1-Alkoxy-3-acyloxy-2-methylpenta-1,3-dienes via Danishefsky-Type Dienes or O-Acylation of Enones
Journal Of Organic Chemistry. 2009.
DOI : 10.1021/jo901878b.
Synthesis of D- and L-erythro 1,5-dithiopent-1-enopyranoside sulfonium salts and their evaluation as glycosidase inhibitors
Tetrahedron-Asymmetry. 2009.
DOI : 10.1016/j.tetasy.2009.07.033.
Ligandless Iron-Catalyzed Desulfinylative C-C Allylation Reactions using Grignard Reagents and Alk-2-enesulfonyl Chlorides
European Journal Of Organic Chemistry. 2009.
DOI : 10.1002/ejoc.200900927.
Chemoselective C-H Bond Activation: Ligand and Solvent Free Iron-Catalyzed Oxidative C-C Cross-Coupling of Tertiary Amines with Terminal Alkynes. Reaction Scope and Mechanism
Organic Letters. 2009.
DOI : 10.1021/ol9002509.
Synthesis and Conformational Analysis of (alpha-D-Galactosyl)phenylmethane and alpha-,beta-Difluoromethane Analogues: Interactions with the Plant Lectin Viscumin
CHEMISTRY - A EUROPEAN JOURNAL. 2009.
DOI : 10.1002/chem.200801394.
A Short and Convenient Synthesis of 1-Deoxymannojirimycin (DMJ) and N-oxy-Analogues from D-Fructose
The Journal of Organic Chemistry. 2009.
DOI : 10.1021/jo802255t.
Palladium-catalyzed desulfinylative C–C allylation of Grignard reagents and enolates using allylsulfonyl chlorides and esters
Tetrahedron. 2009.
DOI : 10.1016/j.tet.2008.11.007.
The prolyl-aminodipeptidases and their inhibitors as therapeutic targets for fibrogenic disorders
Mini Review in Medicinal Chemistry. 2009.
DOI : 10.2174/138955709787316100.
2008
New synthetic seven-membered 1-azasugars displaying potent inhibition towards glycosidases and glucosylceramide transferase
Chembiochem. 2008.
DOI : 10.1002/cbic.200700496.
Quantum calculations on the acid catalyzed rearrangements of norborn-5-en-2-one, 7-oxanorborn-5-en-2-one and 7-azanorborn-5-en-2-one - The electron-releasing effect of homoconjugated carbonyl group
Applied Catalysis A-General. 2008.
DOI : 10.1016/j.apcata.2007.07.048.
Total asymmetric synthesis of glycomimetics and polypropionates of biological interest
Chimia. 2008.
DOI : 10.2533/chimia.2008.519.
Synthesis and L-fucosidase inhibitory potency of a cyclic sugar imine and its pyrrolidine analogue
Tetrahedron-Asymmetry. 2008.
DOI : 10.1016/j.tetasy.2008.06.019.
Iron-Catalyzed Mizoroki–Heck Cross-Coupling Reaction with Styrenes
Advanced Synthesis and Catalysis. 2008.
DOI : 10.1002/adsc.200800662.
Recent Synthetic Approaches Toward Non-anomeric Spiroketals in Natural Products
MOLECULES. 2008.
DOI : 10.3390/molecules13102570.
Iron/copper-catalyzed C–C cross-coupling of aryl iodides with terminal alkynes
Tetrahedron Letters. 2008.
DOI : 10.1016/j.tetlet.2008.07.151.
Functionalized pyrrolidine inhibitors of human alpha- mannosidases II in cancer: optimizing the fit to the active site
Bioorganic and Medicinal Chemistry. 2008.
DOI : 10.1016/j.bmc.2008.06.021.
Spongistatins : biological activity and synthetic studies
Comptes Rendus de l'Académie des Sciences. 2008.
Preparation and synthetic applications of 8-oxabicyclo[3.2.1]oct-6-en-3-one derivatives
Chimia. 2008.
DOI : 10.2533/chimia.2008.221.
Iron-Catalyzed Desulfinylative C-C Cross-Coupling Reactions of Sulfonyl Chlorides with Grignard Reagents
Angewandte Chemie-International Edition. 2008.
DOI : 10.1002/anie.200704858.
2007
Synthesis of monosaccharides and analogues - Part three: Monosaccharides from simple achiral unsaturated compounds
Chimica Oggi-Chemistry Today. 2007.
New efficient route to an advanced precursor of the AB spiroketal of spongistatins
Organic Letters. 2007.
Efficient synthesis of cyclic glycolipids analogues
Synlett. 2007.
DOI : 10.1055/s-2007-973905.
Evaluation of docking programs for predicting binding of Golgi alpha-mannosidase II inhibitors: a comparison with crystallography
PROTEINS-structure, function and bioinformatics. 2007.
2006
Palladium-Catalyzed Desulfitative Mizoroki-Heck Coupling Reactions of Sulfonyl Chlorides with Olefins in a Nitrile-functionalized Ionic Liquid
Synlett. 2006.
DOI : 10.1055/s-2006-944198.
The bora-ene reaction of sulfur dioxide and prop-2-ene-1-boronic esters. New route to sulfoxides
Tetrahedron Letters. 2006.
DOI : 10.1016/j.tetlet.2006.02.071.
Synthesis of new pyrrolidine derivatives as inhibitors of alpha-mannosidase and of glioblastoma cells growth
Heterocycles. 2006.
New efficient synthesis of long chain di- and tri-aminopolyols
European Journal of Organic Chemistry. 2006.
DOI : 10.1002/ejoc.200600276.
Glycosylation pathways as drug targets for cancer: glycosidase inhibitors
Mini Reviews in Medicinal Chemistry. 2006.
DOI : 10.2174/138955706778195162.
Pyrrolidine derivatives as new inhibitors of alpha-mannosidases and growth inhibitors of human cancer cells
Chimia. 2006.
New synthetic route toward polyketide-like macrolides
Synlett. 2006.
DOI : 10.1055/s-2006-932495.
Selective hydrolysis of anti-1,3-diol-acetonides for the differentiation of 1,3-anti and 1,3-syn diols
Tetrahedron Letters. 2006.
DOI : 10.1016/j.tetlet.2005.11.110.
Asymmetric synthesis of the polyol subunit of the polyene macrolide antibiotic RK-397
European journal of organic chemistry. 2006.
DOI : 10.1002/ejoc.200500670.
2005
Noniterative approach to the total asymmetric synthesis of 15-carbon polyketides and analogs with high stereodiversity
Pure and Applied Chemistry. 2005.
DOI : 10.1351/pac200577010131.
Functionalized pyrrolidines as alpha-mannosidase inhibitors and growth inhibitors of human glioblastoma and melanoma cells
Journal of Medicinal Chemistry. 2005.
DOI : 10.1021/jm0409019.
Expeditious asymmetric synthesis of a stereoheptad corresponding to the C(19)-C(27)-ansa chain of rifamycins: Formal total synthesis of Rifamycin S
Chemistry-a European Journal. 2005.
DOI : 10.1002/chem.200400825.
C(1 -> 4)-linked disaccharides through carbonylative Stille cross-coupling
Tetrahedron-Asymmetry. 2005.
Synthesis of aza-C-disaccharides (dideoxyimino-alditols C-linked to monosaccharides) and analogues
Synthesis-Stuttgart. 2005.
Total asymmetric synthesis of (-)-conduramine B-1 and of its enantiomer. N-Benzyl derivatives of conduramine B-1 are beta-glucosidase inhibitors
Bioorganic & Medicinal Chemistry Letters. 2005.
DOI : 10.1016/j.bmcl.2005.04.023.
New 1-amino-1-deoxy- and 2-amino-2-deoxy-polyhydroxyazepanes: synthesis and inhibition of glycosidases
Tetrahedron-Asymmetry. 2005.
Silyl methallylsulfinates: efficient and powerful agents for the chemoselective silylation of alcohols, polyols, phenols and carboxylic acids
Chemical Communications. 2005.
One-pot synthesis of 1-aryl-3-methyl-1,3-dienes using methallyl(trimethyl)silane and aldehydes and their low temperature (Z)->(E) isomerization induced by sulfur dioxide
Tetrahedron. 2005.
DOI : 10.1016/j.tet.2004.11.070.
Palladium-catalyzed desulfitative Mizoroki-Heck couplings of sulfonyl chlorides with mono- and disubstituted olefins: Rhodium-catalyzed desulfitative heck-type reactions under phosphine- and base-free conditions
Chemistry-a European Journal. 2005.
DOI : 10.1002/chem.200400838.
New concise total synthesis of (+)-lentiginosine and some structural analogues
Journal of Organic Chemistry. 2005.
Synthesis of the C(1)-C(11) polyene fragment of apoptolidin with a new sulfur dioxide-based organic chemistry
Chemistry-a European Journal. 2005.
DOI : 10.1002/chem.200500165.
Sulfur dioxide-mediated syntheses of polyfunctional alkenes and (E,Z)- and (E,E)-2,4-dien-1-ones
Organic Letters. 2005.
DOI : 10.1021/ol050006z.
C-linked disaccharide analogue of the Thomsen-Friedenreich (T)-epitope alpha-O-conjugated to L-serine
Chemistry-a European Journal. 2005.
DOI : 10.1002/chem.200401301.
Synthesis and glycosidase inhibitory activity of new penta-substituted C8-glycomimetics
Tetrahedron. 2005.
DOI : 10.1016/j.tet.2005.05.066.
Noniterative approach to the total asymmetric synthesis of 15-carbon polyketides and analogs with high stereodiversity
Pure Appl. Chem.. 2005.
Enzymatic desymmetrization of 1,1 '-methylenedi-[(1R,1 ' S,3R,3 ' S,5S,5 ' R)-3-hydroxy-8-oxabicyclo[3.2.1]-oct-6-ene-1-yl]: Novel precursors of long chain polyketides
Tetrahedron: Asymmetry. 2005.
DOI : 10.1016/j.tetasy.2005.05.038.
2004
First asymmetric synthesis of the cyclohexanone subunit of baconipyrones A and B. Revision of its structure
Organic Letters. 2004.
Synthesis of long-chain polyketide fragments by reaction of 1,3-dioxy-1,3-dienes with allylsilanes: Umpolung with sulfur dioxide
Organic Letters. 2004.
Deracemization of 5-(4-hydroxyphenyl)-5-phenylhydantoin (HPPH): practical synthesis of (-)-(S)-HPPH
Tetrahedron-Asymmetry. 2004.
Synthesis of D- and L-2,3-trans-3,4-cis-4,5-trans-3,4-dihydroxy-5-hydroxymethylproline and tripeptides containing them
Journal of Organic Chemistry. 2004.
DOI : 10.1021/jo049637h.
Non-iterative asymmetric synthesis of C-15 polyketide spiroketals
Helvetica Chimica Acta. 2004.
DOI : 10.1002/hlca.200490136.
The conformational behavior of novel glycosidase inhibitors with substituted azepan structures: An NMR and modeling study
European Journal of Organic Chemistry. 2004.
Polysulfones: Catalysts for alkene isomerization
Angewandte Chemie-International Edition. 2004.
Allyl, methallyl, prenyl, and methylprenyl ethers as protected alcohols: Their selective cleavage with diphenyidisulfone under neutral conditions
Organic Letters. 2004.
DOI : 10.1021/ol049135q.
Polysulfones: solid organic catalysts for the chemoselective cleavage of methyl-substituted allyl ethers under neutral conditions
Chemical Communications. 2004.
Synthesis of N-substituted (3S,4S)- and (3R,4R)-pyrrolidine-3,4-diols: Search for new glycosidase inhibitors
Helvetica Chimica Acta. 2004.
Polyhydroxyazepanes mimicking monosaccharides: Synthesis of an alpha-D-galacto-like iminoheptitol
Heterocycles. 2004.
The first synthesis of substituted azepanes mimicking monosaccharides: a new class of potent glycosidase inhibitors
Organic & Biomolecular Chemistry. 2004.
Palladium-catalyzed conversion of beta,gamma-unsaturated silyl sulfinates into (E)-alkenes: Asymmetric synthesis of polypropionate fragments
Journal of Organic Chemistry. 2004.
Palladium-catalyzed Suzuki-Miyaura cross-couplings of sulfonyl chlorides and boronic acids
Organic Letters. 2004.
DOI : 10.1021/ol036131x.
Palladium-catalyzed desulfitative Sonogashira-Hagihara cross-couplings of arenesulfonyl chlorides and terminal alkynes
Advanced Synthesis & Catalysis. 2004.
Synthesis of C-linked analogues of beta-D-galactopyranosyl-(1 -> 3)-D-galactopyranosides and of beta-D-galactopyranosyl-(1 -> 3)-D-galactal
Tetrahedron-Asymmetry. 2004.
New nonhydrolyzable mimetics of sialyl Lewis x and their binding affinity to P-selectin
Helvetica Chimica Acta. 2004.
DOI : 10.1002/hlca.200490096.
Stereoselective synthesis of novel tetrahydroxypyrrolizidines
Tetrahedron-Asymmetry. 2004.
Sulfur dioxide mediated one-pot, three- and four-component syntheses of polyfunctional sulfonamides and sulfonic esters: Study of the stereoselectivity of the ene reaction of sulfur dioxide
Journal of Organic Chemistry. 2004.
DOI : 10.1021/jo049047j.
Syntheses and glycosidase inhibitory activities of 2-(aminomethyl)-5(hydroxymethyl)pyrrolidine-3,4-diol derivatives
Helvetica Chimica Acta. 2004.
DOI : 10.1002/hlca.200490078.
An expeditious asymmetric synthesis of polyfunctional 1,7-dioxaspiro[5.5]undecanes
European Journal of Organic Chemistry. 2004.
2003
Regioselective rearrangement of 7-azabicyclo[2.2.1]hept-2-aminyl radicals: first synthesis of 2,8-diazabicyclo[3.2.1]oct-2-enes and their conversion into 5-(2-aminoethyl)-2,3,4-trihydroxypyrrolidines, new inhibitors of alpha-mannosidases
Tetrahedron Letters. 2003.
DOI : 10.1016/S0040-4039(03)01141-9.
Efficient resolution of N-Boc-7-azabicyclo[2.2.1]hept-5-en-2-one: formal syntheses of natural epibatidine and its enantiomer
Tetrahedron-Asymmetry. 2003.
Synthesis of enantiomerically pure 1,2-diamine derivatives of 7-azabicyclo[2.2.1]heptane. New leads as glycosidase inhibitors and rigid scaffolds for the preparation of peptide analogues
Journal of Organic Chemistry. 2003.
Synthesis and glycosidase inhibitory activities of 5-(1 ',4 '-dideoxy-1 ',4 '-imino-D-erythrosyl)-2-methyl-3-furoic acid (=5-[3S, 4R)-3,4-dihydroxypyrrolidin-2-yl]-2-methylfuran-3-carboxylic acid) derivitives: New leads as selective alpha-L-fucosidase and beta-galactosidase inhibitors
Helvetica Chimica Acta. 2003.
DOI : 10.1002/hlca.200390152.
Equilibrium and kinetic deuterium isotope effects on the hetero-Diels-Alder addition of sulfur dioxide
Angewandte Chemie-International Edition. 2003.
Scope and limitations of the double [4+3]-cycloadditions of 2-oxyallyl cations to 2,2 '-methylenedifuran and derivatives
Journal of Organic Chemistry. 2003.
DOI : 10.1021/jo020678s.
The hetero-Diels-Alder addition of sulfur dioxide: The pseudo-chair conformation of a 4,5-dialkylsultine
Chemistry-a European Journal. 2003.
DOI : 10.1002/chem.200304932.
Palladium-catalyzed stille cross-couplings of sulfonyl chlorides and organostannanes
Journal of the American Chemical Society. 2003.
DOI : 10.1021/ja038328q.
Syntheses of beta-C(1 -> 3)-Glucopyranosides of 2-and 4-deoxy-D-hexoses
Helvetica Chimica Acta. 2003.
DOI : 10.1002/hlca.200390037.
Synthesis and glycosidase inhibitory activity of 7-deoxycasuarine
Helvetica Chimica Acta. 2003.
DOI : 10.1002/hlca.200390248.
Stereoselective syntheses of 1,4-dideoxy-1,4-imino-octitols and novel tetrahydroxyindolizidines
Journal of Organic Chemistry. 2003.
Synthesis and alpha-mannosidase inhibitory evaluation of (2R,3R,4S)- and (2S,3R,4S)-2-(aminomethyl)pyrrolidine-3,4-diol derivatives
Helvetica Chimica Acta. 2003.
DOI : 10.1002/hlca.200390153.
An expeditious, non-iterative, and asymmetric synthesis of 3,5,7,9,11,13,15-heptahydroxypentadecanals
European Journal of Organic Chemistry. 2003.
Synthesis and glycosidase inhibitory activities of 2-(aminoalkyl)pyrrolidine-3,4-diol derivatives
Bioorganic & Medicinal Chemistry. 2003.
2002
Synthesis of 2,2 ',2 '',2 '''-(1,2-ethanediylidene)tetrafuran and Diels-Alder reaction with dimethyl acetylenedicarboxylate
Heterocycles. 2002.
Synthesis of 1,2,3,4-tetrahydro-1,2-dimethylidenenaphthalene: A reactive s-cis-butadiene undergoing highly chemo- and regioselective cyclodimerization
Helvetica Chimica Acta. 2002.
Competition between hetero-Diels-Alder and cheletropic additions of sulfur dioxide to 2-substituted buta-1,3-dienes. Synthesis of 2-(1-naphthyl)and 2-(2-naphthyl)buta-1,3-diene
Helvetica Chimica Acta. 2002.
The hetero-Diels-Alder addition of sulfur dioxide to 1-fluorobuta-1,3-dienes: The sofa conformations preferred by 6-fluorosultines (6-fluoro-3,6-dihydro-1,2-oxathiin-2-oxides) enjoy enthalpic and conformational anomeric effects
Chemistry-a European Journal. 2002.
DOI : 10.1002/1521-3765(20020315)8:6<1336::AID-CHEM1336>3.0.CO;2-R.
Substituent effect on the competition between hetero-Diels-Alder and cheletropic additions of sulfur dioxide to 1-substituted buta-1,3-dienes
Helvetica Chimica Acta. 2002.
The synthesis of disaccharides, oligosaccharides and analogues containing thiosugars
Current Organic Chemistry. 2002.
DOI : 10.2174/1385272024604952.
Synthesis of a new C(1 -> 2)-linked iminodisaccharide starting from levoglucosenone
Helvetica Chimica Acta. 2002.
DOI : 10.1002/1522-2675(200201)85:1<152::AID-HLCA152>3.0.CO;2-L.
One-pot, asymmetric and diastereoselective four-component synthesis of polyfunctional (Z)-alkenyl methyl sulfones with three stereogenic centers
Helvetica Chimica Acta. 2002.
DOI : 10.1002/1522-2675(200206)85:6<1674::AID-HLCA1674>3.0.CO;2-2.
Synthesis of [(2S,3S,4R)-3,4-dihydroxypyrrolidin-2-yl]-5-methylfuran-4-carboxylic acid derivatives: New leads as selective beta-galactosidase inhibitors
Bioorganic & Medicinal Chemistry Letters. 2002.
DOI : 10.1016/S0960-894X(02)00397-9.
Hetero-Diels-Alder and cheletropic additions of sulfur dioxide to 1,2-dimethylidenecycloalkanes. Determination of thermochemical and kinetics parameters for reactions in solution and comparison with estimates from quantum calculations
Helvetica Chimica Acta. 2002.
DOI : 10.1002/1522-2675(200203)85:3<712::AID-HLCA712>3.0.CO;2-5.
Ab initio and experimental studies on the hetero-Diels-Alder and cheletropic additions of sulfur dioxide to (E)-1-methoxybutadiene: A mechanism involving three molecules of SO2
Journal of Organic Chemistry. 2002.
DOI : 10.1021/jo010998w.
Synthesis of (1 -> 3)-C and homo(1 -> 3)-C-linked iminodisaccharides starting from levoglucosenone and isolevoglucosenone
Heterocycles. 2002.
One-pot, four-component synthesis of polyfunctional sulfones
Synthesis-Stuttgart. 2002.
One-pot, three-component synthesis of open-chain, polyfunctional sulfones
Synthesis-Stuttgart. 2002.
Synthesis of seven- and eight-membered carbasugar analogs via ring-closing metathesis and their inhibitory activities toward glycosidases
Tetrahedron-Asymmetry. 2002.
Total asymmetric synthesis of a new 9,12-anhydroerythronolide aglycone
Helvetica Chimica Acta. 2002.
DOI : 10.1002/1522-2675(200202)85:2<417::AID-HLCA417>3.0.CO;2-1.
An efficient combinatorial method for the discovery of glycosidase inhibitors
Chembiochem. 2002.
DOI : 10.1002/1439-7633(20020503)3:5<466::AID-CBIC466>3.0.CO;2-D.
Asymmetric synthesis of 1-aminopentadecane-3,5,7,9,11,13,15-heptols and of 1,15-diaminopentadecane-3,5,7,9,11,13-hexols and derivatives
Synthesis. 2002.
Synthesis of tri-and tetramines containing two 2,3-dihydroxypyrrolidine moieties and their inhibitory activity toward alpha-mannosidases
Arkivoc. 2002.
2001
Derivatives of (2R,3R,4S)-2-Aminomethylpyrrolidine-3,4-diol are Selective alpha-Mannosidase Inhibitors
Bioorganic and Medicinal Chemistry Letters. 2001.
Synthesis of a (2R,6R)-2-(hydroxymethyl)-6-propa-1,2-dienyl-2H-pyran-3(6H)-one derivative, a new enone for the convergent construction of C-glycosides of D-disaccharides
Synlett. 2001.
Synthesis of a C-disaccharide analog of the Thomsen-Friedenreich (T) epitope
Synlett. 2001.
Monosaccharide and disaccharide mimics: New molecular tools for biology and medicine
Chimia. 2001.
Synthesis of the C-disaccharide alpha-C(1 -> 3)-L-fucopyranoside of N-acetylgalactosamine
Journal of Carbohydrate Chemistry. 2001.
From 2,2 '-methylenedifuran to all stereomeric pentadecane-1,3,5,7,9,11,13,15-octols
Journal of Organic Chemistry. 2001.
DOI : 10.1021/jo010172u.
The hetero-Diels-Alder addition of sulfur dioxide: structure of the first crystalline sultine. Quantum calculations on the conformations of 6-fluoro-3,6-dihydro-1,2-oxathiine 2-oxides
Chemical Communications. 2001.
Synthesis and biological properties of monothiosaccharides
Current Organic Chemistry. 2001.
DOI : 10.2174/1385272013374743.
New leads for selective inhibitors of alpha-L-fucosidases. Synthesis and glycosidase inhibitory activities of [(2R,3S,4R)-3,4-dihydroxypyrrolidin-2-yl]furan derivatives
Bioorganic & Medicinal Chemistry Letters. 2001.
DOI : 10.1016/S0960-894X(01)00497-8.
Development of a new carbon-carbon bond forming reaction. New organic chemistry of sulfur dioxide. Asymmetric four-component synthesis of polyfunctional sulfones
Journal of Organic Chemistry. 2001.
DOI : 10.1021/jo0101712.
Four component synthesis of (Z)-4-alkoxy-1,3-dimethylalk-2-enyl methyl sulfones: on the intermediacy of sultines (3,6-dihydro-1,2-oxathiin-2-oxides) arising from suprafacial hetero-Diels-Alder additions of sulfur dioxide
Tetrahedron Letters. 2001.
DOI : 10.1016/S0040-4039(00)02102-X.
alpha- and beta-homogalactonojirimycins (alpha- and beta-homogalactostatins): Synthesis and further biological evaluation
Bioorganic & Medicinal Chemistry. 2001.
DOI : 10.1016/S0968-0896(00)00343-6.
Asymmetric synthesis of complicated bicyclic and tricyclic polypropanoates via the double Diels-Alder addition of 2,2 '-ethyiidenebis[3,5-dimethylfuran]
Helvetica Chimica Acta. 2001.
DOI : 10.1002/1522-2675(20010228)84:2<431::AID-HLCA431>3.0.CO;2-W.
Amino(hydroxymethyl)cyclopen-tanetriols, an emerging class of potent glycosidase inhibitors - Part I: Synthesis and evaluation of beta-D-pyranoside analogues in the manno, gluco, galacto, and GlcNAc series
Chembiochem. 2001.
DOI : 10.1002/1439-7633(20010504)2:5<365::AID-CBIC365>3.0.CO;2-M.
Recent progress in the synthesis of zaragozic acids and analogs
Current Organic Chemistry. 2001.
DOI : 10.2174/1385272013375328.
Synthesis and solution conformational analysis of 2,3-anhydro-3-C-[(1R)-2,6-anhydro-1-deoxy-1-fluoro-D-glycero-D-gulo-hept itol-1-C-yl]-beta-D-gulo-furanose: First example of a monofluoromethylene-linked C-disaccharide
Journal of Organic Chemistry. 2001.
DOI : 10.1021/jo0102462.
Stereoselective synthesis of 8-oxabicyclo[3.2.1]octane-2,3,4,6,7-pentols and total asymmetric synthesis of 2,6-anhydrohepturonic acid derivatives and of beta-C-manno-pyranosides suitable for the construction of (1 -> 3)-C,C-linked trisaccharides
Helvetica Chimica Acta. 2001.
DOI : 10.1002/1522-2675(20010613)84:6<1363::AID-HLCA1363>3.0.CO;2-M.
Stereoselective synthesis of new 8-oxabicyclo[3.2.1]oct-6-en-2-one and 8-oxabicyclo[3.2.1]octa-3,6-dien-2-one derivatives. The electron-releasing and electron-withdrawing effects of homoconjugated ketones
Indian Journal of Chemistry Section B-Organic Chemistry Including Medicinal Chemistry. 2001.
2000
Synthesis of a C29-C51 Subunit of Spongistatin 1 (Altohyrtin A) Starting from (R)-3-Benzyloxy-2-methylpropan-1-ol
Journal of Organic Chemistry. 2000.
DOI : 10.1021/jo991642b.
Convergent syntheses of C(1 -> 3)-linked disaccharides starting from isolevoglucosenone
Tetrahedron-Asymmetry. 2000.
Sugar mimetics: Why and how
Chimia. 2000.
Synthesis of rare carbohydrates and analogues starting from enantiomerically pure 7-oxabicyclo[2.2.1]heptyl derivatives ("naked sugars")
Current Organic Chemistry. 2000.
DOI : 10.2174/1385272003376175.
A new, non-iterative asymmetric synthesis of long-chain 1,3-polyols
Chemistry-a European Journal. 2000.
Asymmetric syntheses of new polyhydroxylated quinolizidines: Cross-aldol reactions of 7-oxabicyclo[2.2.1]heptan-2-one and 3a,4a,7a,7b-tetrahydro[1,3]dioxolo[4,5]furo[2,3-d]isoxazole-3-carbaldehy de derivatives
Helvetica Chimica Acta. 2000.
O-17 NMR spectroscopy of sulfolenes (2,5-dihydrothiophene-1,1-dioxides) and sultines (3,6-dihydro-1,2-oxathiin-2-oxides)-experiment and quantum calculations: Synthesis of 4,9-dioxo-1,2-oxathiacyclodecane-2-oxide, a new heterocycle
Chemistry-a European Journal. 2000.
DOI : 10.1002/(SICI)1521-3765(20000515)6:10<1858::AID-CHEM1858>3.0.CO;2-U.
The C-disaccharide alpha-C(1 -> 3)-mannopyranoside of N-acetylgalactosamine is an inhibitor of glycohydrolases and of human alpha-1,3-fucosyltransferase VI. its epimer alpha-(1 -> 3)-mannopyranoside of N-acetyltalosamine is not
Journal of Organic Chemistry. 2000.
DOI : 10.1021/jo991952u.
A new asymmetric carbon-carbon bond forming reaction: Four-component stereoselective synthesis of (Z)-4,6-dihydroxy-3-methylalk-2-enyl methyl sulfones
Angewandte Chemie-International Edition. 2000.
Oxetane formation by 1,3-migration of benzyloxy group in 7-oxabicyclo[2.2.1]hept-2-yl cations: Synthesis of 4,7-dioxatricyclo[3.2.1.O-3,O-6]octane and 2-oxabicyclo[2.2.2]octane encrusted in the 1,4 : 5,8-diepoxy-perhydrophenanthrene ring system
Heterocycles. 2000.
Asymmetric synthesis of polycyclic polyketides via the double Diels-Alder addition of 2,2 '-ethylidenebis[3,5-dimethylfuran]
Synlett. 2000.
Synthesis of 1,1 '-methylenedi[(1R,1 ' R,3R,3 ' R,5R,5 ' R)-8-oxabicyclo[3.2.1]oct-6-en-3-ol] and derivatives: precursors of long-chain polyketides
Tetrahedron-Asymmetry. 2000.
Total synthesis of a protected form of 2,6-anhydro-5-azido-3,5-dideoxy-2-C-hydroxymethyl-L-allo-heptose; a potential precursor of analogs of C-glycosides of neuraminic acid
Tetrahedron-Asymmetry. 2000.
Synthesis of (Z)-3-deoxy-3-(1,2,3,6-tetradeoxy-3,6-imino-L-arabino-hexitol-1-C-yliden e)-D-xylo-hexose derivatives. First examples of homo-(1 -> 3)-C-linked iminodisaccharides
Journal of Carbohydrate Chemistry. 2000.
Polyhydroxypyrrolidine glycosidase inhibitors related to (+)-lentiginosine
Journal of Carbohydrate Chemistry. 2000.
1999
Short and convergent synthesis of (1 -> 3)-C-linked imino disaccharides (aza-C-disaccharides)
Journal of Organic Chemistry. 1999.
Convergent synthesis of (1 -> 2)- and (1 -> 4)-C-linked imino disaccharides
Chemical Communications. 1999.
Derivatives of 7-oxabicyclo[2.2.1]heptane in nature and as useful synthetic intermediates
Tetrahedron. 1999.
DOI : 10.1016/S0040-4020(99)00845-5.
Synthesis of a polyhydroxyquinolizidine bearing a polyhydroxylated carbon side-chain
Synlett. 1999.
Specific, uncompetitive inhibition of beta-galactosidases by a 5,6-isopropylidenedioxyfuro[2,3-d]isoxazole-3-methanol derivative
Bioorganic & Medicinal Chemistry Letters. 1999.
DOI : 10.1016/S0960-894X(98)00722-7.
Synthesis of alpha-C(1 -> 3)-mannopyranoside of N-acetylgalactosamine, a new beta-galactosidase inhibitor
Bioorganic & Medicinal Chemistry Letters. 1999.
DOI : 10.1016/S0960-894X(99)00064-5.
Stereoselective synthesis of 5a-ethyl-1,2,3,3a,4,5,5a,6,9a,9b-decahydro-1,3,4-trihydroxy-3a-(hydroxym ethyl)-7H-benz[e]inden-7-one derivatives
Helvetica Chimica Acta. 1999.
DOI : 10.1002/(SICI)1522-2675(19990908)82:9<1371::AID-HLCA1371>3.0.CO;2-N.
Polyhydroxylated perhydro-1H-benz[e]indenyl derivatives with two angular 3a,5a-carbaldehyde moieties
Synlett. 1999.
Total, asymmetric synthesis of methyl 3-deoxy-3-(1 ',2 ',6 '-trideoxy-2 ',6 '-imino-D-galactitol-1-yl)-alpha-D-manno-pyranoside (A C-linked imino disaccharide): Conformational analysis and glycosidase inhibition
Synthesis. 1999.
DOI : 10.1055/s-1999-3645.
A short and flexible route to aza-beta-(1 -> 6)-C-disaccharides: Selective alpha-glycosidase inhibitors
European Journal of Organic Chemistry. 1999.
Total asymmetric synthesis of doubly branched carba-hexopyranoses and amino derivatives starting from the Diels-Alder adducts of maleic anhydride to furfuryl esters
Helvetica Chimica Acta. 1999.
DOI : 10.1002/(SICI)1522-2675(19990609)82:6<821::AID-HLCA821>3.0.CO;2-K.
En route toward squalestatins and analogues from furfuryl alcohol and maleic anhydride
Tetrahedron Letters. 1999.
DOI : 10.1016/S0040-4039(99)01068-0.
Synthesis of a 5-hydroxypiperidine-2,3,4,6-tetramethanol, a new 2,6-dideoxy-2,6-iminoheptitol derivative
Journal of Organic Chemistry. 1999.
DOI : 10.1021/jo991228b.
Regioselective base-induced ethereal bridge openings of 7-oxabicyclo[2.2.1]heptane-2,3-dicarboxylic derivatives; Synthesis of squalestatin core analogues
Synlett. 1999.
Total stereoselective syntheses of beta-C-manno-pyranosides and of beta-C(1 -> 3)-linked disaccharides
Tetrahedron Letters. 1999.
DOI : 10.1016/S0040-4039(99)00432-3.
Resolution of 7-oxabicyclo[2.2.1]hept-5-en-2-one via cyclic aminals
Tetrahedron-Asymmetry. 1999.
Migratory insertion reactions of norbornene, norbornadiene and 7-oxanorbornene derivatives into the palladium-carbon bond of heterodinuclear Fe-Pd-Acyl complexes. Substrate influence on the Pd coordination sphere and crystal structure of [(OC)(3)Fe{mu-Si(OMe)(2)(OMe)}(mu-dppa)Pd{C9H9NO3C(=O)Me}]
New Journal of Chemistry. 1999.
DOI : 10.1039/a905842g.
Total, asymmetric synthesis of ethyl D-ido-4-heptulosuronate derivatives starting from diethyl 4-oxopimelate
Tetrahedron: Asymmetry. 1999.
DOI : 10.1016/S0957-4166(99)00120-2.
1998
Short, stereoselective syntheses of C(1 -> 3)-linked disaccharides
Tetrahedron Letters. 1998.
Combinatorial Diels-Alder approach to the synthesis of anti-tumor anthracyclines and analogues
Current Organic Chemistry. 1998.
Synthesis of 4-hydroxy-2,6-bis(hydroxymethyl)tetrahydropyran-2-carbaldehyde derivatives
Synlett. 1998.
Total syntheses of (+)- and (-)-1-deoxynojirimycin (1,5-dideoxy-1,5-imino-D- and L-glucitol) and of (+)- and (-)-1-deoxyidonojirimycin (1,5-dideoxy-1,5-imino-D- and L-iditol) via furoisoxazoline-3-aldehydes
Carbohydrate Research. 1998.
DOI : 10.1016/S0008-6215(98)00287-0.
5a-carba-beta-D-, 5a-carba-beta-L- and 5-thio-beta-L-xylopyranosides as new orally active venous antithrombotic agents
Helvetica Chimica Acta. 1998.
DOI : 10.1002/(SICI)1522-2675(19981111)81:11<2043::AID-HLCA2043>3.0.CO;2-6.
Synthesis of C-linked imino disaccharides (=aza-C-disaccharides) with a pyrrolidine-3,4-diol moiety attached at C(3) of galactose via a hydroxymethylene linker and of a 7-(1,2,3-trihydroxypropyl)-octahydroxyindolizine-1,2,6,8-tetrol
Helvetica Chimica Acta. 1998.
DOI : 10.1002/hlca.19980810552.
Stereoselective synthesis of new conduramines and aminocyclitol derivatives
Synlett. 1998.
Carbaxylosides of 4-ethyl-2-oxo-2H-benzopyran-7-yl as non-hydrolyzable, orally active venous antithrombotic agents
Bioorganic & Medicinal Chemistry Letters. 1998.
DOI : 10.1016/S0960-894X(98)00283-2.
Competition between hetero-Diels-Alder and cheletropic addition of sulfur dioxide. Theoretical and experimental substituent effects on the relative stability of 3,6-dihydro-1,2-oxathiin-2-oxides (sultines) and 2,5-dihydrothiophene-1,1-dioxides (sulfolenes). Anomeric effects in sultine and 6-substituted derivatives
Journal of Organic Chemistry. 1998.
Sulfur dioxide promotes its hetero-Diels-Alder and cheletropic additions to 1,2-dimethylidenecyclohexane
Journal of the American Chemical Society. 1998.
Total asymmetric synthesis of seco-acids of 9,12-anhydroerythronolide aglycons
Tetrahedron Letters. 1998.
DOI : 10.1016/S0040-4039(98)00691-1.
Total synthesis of the C-37-C-45 F-ring fragment of spongistatins
Tetrahedron Lett.. 1998.
1997
Synthesis of peptides using palladium promoted selective removal of allyloxycarbonyl protecting groups in aqueous medium
Tetrahedron Letters. 1997.
DOI : 10.1016/S0040-4039(97)00535-2.
Chemoselective Removal of Allylic Protecting Groups Using Water-Soluble Pd(OAc)2/TPPTS Catalyst
Journal of Molecular Catalysis A: Chemical. 1997.
The electron-releasing carbonyl group .1. Discovery and theoretical studies
Chimica Oggi-Chemistry Today. 1997.
The electron-releasing carbonyl group .2. Spectroscopic detection and synthetic applications
Chimica Oggi-Chemistry Today. 1997.
Remote control of Diels-Alder additions. Enantioselective synthesis of (2R)-1,2,3,4-tetrahydro-2-hydroxy-5,8-dimethoxynaphthalen-2-yl methyl ketone (Wong's anthracycline intermediate) from furfural
Tetrahedron-Asymmetry. 1997.
Tandem oxyallylations and retro-ene eliminations. One pot stereoselective synthesis of polypropionate fragments with three contiguous stereogenic centers and one (E)-alkene unit
Tetrahedron Letters. 1997.
Highly stereoselective synthesis of perhydro-8a-(hydroxymethyl)phenanthrene-1,2,4,5,7,8-hexol and derivatives
Journal of Organic Chemistry. 1997.
DOI : 10.1021/jo962331t.
Dihydroxypyrrolidines C-linked to galactose. Total synthesis of a specific inhibitor of alpha-mannosidases
Bioorganic & Medicinal Chemistry Letters. 1997.
DOI : 10.1016/S0960-894X(97)00135-2.
Long-distance effect on one-bond C-C scalar couplings upon introduction of a double bond in bicyclic systems
Helvetica Chimica Acta. 1997.
DOI : 10.1002/hlca.19970800105.
C-glycosides and C-disaccharide precursors through carbonylative Stille coupling reactions
Tetrahedron Letters. 1997.
DOI : 10.1016/S0040-4039(96)02367-2.
New carbon-carbon bond formation through oxyallylation of enoxysilanes with sulfur dioxide adduct of 1-methoxybutadiene. Stereoselective synthesis of (Z)-4-methoxy-6-oxoalk-2-enyl methyl sulfones
Tetrahedron Letters. 1997.
High-performance liquid chromatography of the renal blood flow marker p-aminohippuric acid (PAH) and its metabolite N-acetyl PAH improves PAH clearance measurements
Journal of Chromatography B. 1997.
DOI : 10.1016/S0378-4347(97)00396-4.
Aza-C-disaccharides: Synthesis of 6-deoxygalactonojirimycin beta-C(1->3) linked with D-altrofuranosides and D-galactose
Journal of Organic Chemistry. 1997.
DOI : 10.1021/jo970151t.
1996
Intramolecular Heck-type Reactions in Aqueous Medium. A Dramatic Change in Regioselectivity
Tetrahedron Letters. 1996.
DOI : 10.1016/0040-4039(96)00253-5.
'Naked sugars of the second generation': Asymmetric synthesis of long-chain polypropionates and analogues starting with acetone
Pure and Applied Chemistry. 1996.
Remote substituent control of the regioselectivity of the aryl- and vinylpalladation of 7-oxabicyclo[2.2.1]heptenes
Tetrahedron Letters. 1996.
DOI : 10.1016/0040-4039(96)00237-7.
The simultaneous double Diels-Alder addition of 1,1-bis(3,5-dimethylfur-2-yl)ethane; Toward a new, asymmetric synthesis of long-chain polypropionate fragments and analogues
Tetrahedron Letters. 1996.
DOI : 10.1016/0040-4039(96)00771-X.
Total asymmetric synthesis of long-chain, branched carbohydrates and of an aza-C-disaccharide
Tetrahedron Letters. 1996.
DOI : 10.1016/0040-4039(96)00189-X.
Stereoselective synthesis of alpha-C-galactopyranosides of conduritols and aminoconduritols
Synlett. 1996.
Synthesis of beta-D-(1->3)-C-linked 1,5,6-trideoxy-1,5-iminogalactoside of D-altrose derivatives
Tetrahedron Letters. 1996.
DOI : 10.1016/0040-4039(95)02214-7.
Synthesis of (+)-3,7,8-trideoxy-3,7-imino-D-threo-L-galacto-octitol and its inhibition of beta-glucosidases
Carbohydrate Research. 1996.
DOI : 10.1016/0008-6215(95)00348-7.
A new strategy for the synthesis of selectively protected spermidine and norspermidine derivatives
Synlett. 1996.
1995
Pi-Allyl Palladium Methodology for Selective Deprotection of Allylamines. Practical Synthesis of Secondary Amines
Bulletin de la société chimique de France. 1995.
Competition between Cheletropic and Homocheletropic Additions of Sulfur-Dioxide to 2,3,5,6-Tetrakis(Methylene)Bicyclo[2.2,N]Alkanes - Crystal and Molecular-Structures of 2 3-Thiabicyclo[3.1.0]Hexane 3,3-Dioxide Derivatives
Tetrahedron. 1995.
DOI : 10.1016/0040-4020(94)01035-X.
Remote Substituent Effect on the Electrophilic Additions of 1,3-Dienes - Synthesis of (2r)-5-(Acetoxymethyl)-2-Acetyl-1,2,3,4-Tetrahydro-10-Methoxynaphthacene -2,12-Diyl Diacetate
Tetrahedron. 1995.
DOI : 10.1016/0040-4020(95)00317-2.
Stereoselective Syntheses of Branched-Chain Carbohydrates Bearing Furan and Pyrrole Moieties
Tetrahedron Letters. 1995.
DOI : 10.1016/0040-4039(95)01849-D.
Synthesis of Polypropionate Fragments Containing Tertiary-Alcohol Moieties - Cross-Aldolisations with Lithium Enolates of 7-Oxabicyclo[2.2.1]Heptan-2-One Derivatives
Helvetica Chimica Acta. 1995.
DOI : 10.1002/hlca.19950780205.
Synthesis of an Alpha-C-Galactoside of a Carbasugar - a New Class of Disaccharide Mimics
Tetrahedron Letters. 1995.
DOI : 10.1016/0040-4039(95)00548-Q.
Regioselective Synthesis of 5-Endo,6-Endo-Dihydroxy-7-Oxabicyclo[2.2.1]Heptan-2-One with Differential Protection of the Diol Group
Synlett. 1995.
Synthesis of Undeculofuranoside Derivatives of the Herbicidins and of Analogs
Journal of Organic Chemistry. 1995.
DOI : 10.1021/jo00123a021.
Synthesis of (-)-6-(3'-Aminopropyloxy)Methyl-4-Demethoxy-6,7-Dideoxy-Daunomycinon, a New DNA Intercalator Related to Anthracyclines
Bioorganic & Medicinal Chemistry Letters. 1995.
DOI : 10.1016/0960-894X(95)00070-A.
Reductive oxa ring opening of 7-oxabicyclo[2.2.1]heptan-2-ones. Synthesis of C-alpha-galactosides of carbapentopyranoses
Journal of Organic Chemistry. 1995.
DOI : 10.1021/jo00131a007.
Assignment of the Absolute-Configuration of Natural Lentiginosine by Synthesis and Enzymatic Assays of Optically Pure (+)-Enantiomers and (-)-Enantiomers
Journal of Organic Chemistry. 1995.
DOI : 10.1021/jo00126a033.
Stereoselective Synthesis of 2,4,6-Trimethylcyclohex-4-Ene-1,3-Diol Derivatives and of Polypropionate Fragments with 4 Contiguous Stereogenic Centers
Helvetica Chimica Acta. 1995.
DOI : 10.1002/hlca.19950780206.
SELECTIVE DEPROTECTION OF ALLYL AMINES USING PALLADIUM
Tetrahedron Letters. 1995.
New Synthetic Applications of Water Acetate Pd/TPPTS Catalyst Generated in situ. Evidence for true Pd(0) Valent Species Intermediate
Journal of Organic Chemistry. 1995.
1994
Selective Deprotection Method Using Palladium Water Soluble Catalysts
Tetrahedron Letters. 1994.
A New Stereoselective and Convergent Approach to the Synthesis of Long-Chain Polypropionate Fragments
Journal of Organic Chemistry. 1994.
DOI : 10.1021/jo00099a020.
Remote Substituent Effects on the Cheletropic and Homocheletropic Additions of Sulfur-Dioxide to Exocyclic Polyenes Grafted onto Bicyclo[2.2.2]Octane Skeletons
Bulletin De La Société Chimique De France. 1994.
Homocheletropic Addition of Sulfur-Dioxide to 1,4-Dienes - Competition between Cheletropic and Homocheletropic Additions of Polyenes
Journal of the American Chemical Society. 1994.
DOI : 10.1021/ja00087a076.
Pi-Facial Diastereoselection in [4+2]-Cycloadditions of 3,4-Epoxy-2-Methyleneoxolanes with Oxadienes - a Short Synthesis of Spiroketals
Tetrahedron. 1994.
DOI : 10.1016/S0040-4020(01)85288-1.
Face Selectivity of the Diels-Alder Additions and Cheletropic Additions of Sulfur-Dioxide to 2-Vinyl-7-Oxabicyclo[2.2.1]Hept-2-Ene Derivatives
Helvetica Chimica Acta. 1994.
DOI : 10.1002/hlca.19940770326.
Homochiral Matching in the Diels-Alder Clyclodimerization 2-Vinyl-7-Oxabicyclo[2.2.1]Hept-2-Ene Derivatives
Tetrahedron Letters. 1994.
DOI : 10.1016/0040-4039(94)88176-6.
Enantiomerically Pure 7-Oxabicyclo(2.2.1)Hept-5-En-2-Yl Derivatives (Naked Sugars) as Synthetic Intermediates .25. Total Asymmetric-Synthesis of 3-Amino-3-Deoxy-L-Talose and Derivatives
Carbohydrate Research. 1994.
Photoreductive Changes of Phenyl-Selenium Bonds of Phenylselenoalkanes
Tetrahedron Letters. 1994.
DOI : 10.1016/0040-4039(94)88021-2.
Naked Sugars as Synthetic Intermediates .26. Synthesis of Alpha-D-(1-]3) and Alpha-D-(1-]4)-C-Linked Galactosides of D-Mannose Derivatives - Conformation of Alpha-C-Galactosides
Tetrahedron-Asymmetry. 1994.
Total Asymmetric-Synthesis of 5-Deoxy-5-Thio-L-Allose
Journal of Carbohydrate Chemistry. 1994.
Total Asymmetric Syntheses of 1,5-Dideoxy-1,5-Iminooctitols and 1,2,6,7,8-Pentahydroxyindolizidines
Journal of Organic Chemistry. 1994.
Polypropionate Fragments with 4 Contiguous Chiral Centers from Acetone
Tetrahedron Letters. 1994.
DOI : 10.1016/S0040-4039(00)77066-3.
Asymmetric Total Synthesis of (11r,12s,13s,9z,15z)-9,12,13-Trihydroxyoctadeca-9,15-Dienoic Acid, a Self-Defensive Agent against Rice-Blast Disease
Helvetica Chimica Acta. 1994.
DOI : 10.1002/hlca.19940770605.
Syntheses of Stable Alpha-Silyloxyepoxides and Alpha-Chloroalkyl Silyl Ethers Derivatives of 3,10-Dioxa-5-Azatricyclo[5.2.1.0/2,6]Dec-4-Enes
Synthetic Communications. 1994.
Unexpected Selectivity between Pinacolic Rearrangement and Intramolecular Displacement in the Acid-Promoted Epoxide Ring-Opening of 6-Exo-Cyano-3,8-Dioxabicyclo[3.2.1.0(2,4)]Oct-6-Endo-Yl Esters
Tetrahedron. 1994.
DOI : 10.1016/S0040-4020(01)86963-5.
Enantioselective Synthesis of (-)-Conduramine C-1 and Aminobromocyclitol Derivatives
Helvetica Chimica Acta. 1994.
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1993
Practical Palladium-Mediated Deprotective Method of Allyloxycarbonyl Groups in Aqueous Media
Tetrahedron. 1993.
A General and Simple Removal of Allyloxycarbonyl Protecting Group by Palladium-Mediated Reactions Using Nitrogen and Sulfur Nucleophiles
Synlett. 1993.
DOI : 10.1055/s-1993-22570.
2,3,5,6-Tetrakis(Methylene)-1,4-Cyclohexanediyl (1,2,4,5-Tetramethylenebenzene), a Disjoint Non-Kekule Singlet Hydrocarbon Biradical
Journal of the American Chemical Society. 1993.
DOI : 10.1021/ja00071a020.
Syntheses of Exo-3,8-Dioxatricylo[3.2.1.0(2,4)]Octane and 4,7-Dioxatricyclo[3.2.1.0(3,6)]Octane and the Relative Basicities of Their Ethereal Moieties
Journal of Organic Chemistry. 1993.
Total Asymmetric-Synthesis of Polypropionate Fragments and Doubly Branched Heptono-1,4-Lactones
Tetrahedron Letters. 1993.
DOI : 10.1016/S0040-4039(00)60444-6.
The Homoconjugated Electron-Releasing Carbonyl Group of 1-Methylbicyclo[2.2.1]Hept-5-En-2-One - Regioselective Syntheses of 5-Chloro-1-Methylbicyclo[2.2.1]Hept-5-En-2-One and 6-Chloro-1-Methylbicyclo[2.2.1]Hept-5-En-2-One
Helvetica Chimica Acta. 1993.
DOI : 10.1002/hlca.19930760619.
Pi-Facial Diastereoselectivity in the Electrophilic and Electrophilic Nucleophilic Additions to Dimethyl (1r,2r,3s,4s)-Bicyclo[2.2.2]Oct-5-Ene-2,3-Dicarboxylate
Journal of the Chemical Society, Chemical Communications. 1993.
Highly Stereoselective, Total Synthesis of Beta-C-Hexopyranosyl Derivatives
Tetrahedron Letters. 1993.
DOI : 10.1016/S0040-4039(00)77480-6.
The Demjanov and Tiffeneau-Demjanov One-Carbon Ring Enlargements of 2-Aminomethyl-7-Oxabicyclo[2.2.1]Heptane Derivatives - the Stereoselective and Regioselective Additions of 8-Oxabicyclo[3.2.1]Oct-6-En-2-One to Soft Electrophiles
Tetrahedron. 1993.
DOI : 10.1016/S0040-4020(01)80352-5.
Total Synthesis of Undeculofuranosiduronic Acid-Derivatives Related to Herbicidins
Tetrahedron Letters. 1993.
DOI : 10.1016/S0040-4039(00)60529-4.
Total Synthesis of the Gastroprotective Substance Ai-77-B and of Analogs
Helvetica Chimica Acta. 1993.
Enantioselective Synthesis of (R)-(-)-2-Acetyl-2,5,12-Trihydro-1,2,3,4-Tetrahydro-6,11-Naphthacenequin One Via Diastereoselective Diels-Alder Cycloaddition
Tetrahedron Letters. 1993.
DOI : 10.1016/S0040-4039(00)77479-X.
Site Selectivity and Regioselectivity of the Hetero-Diels-Alder and Cheletropic Additions of Sulfur-Dioxide to a 2,3,6,7-Tetramethylidenebicyclo[3.2.1]Octane Derivative
Tetrahedron Letters. 1993.
DOI : 10.1016/S0040-4039(00)73728-2.
Stabilizing Effect by Geminal Dioxy Substitution and Anomeric Effect in 3,6-Dihydro-6-Methoxy-1,2-Oxathiin 2-Oxides
Helvetica Chimica Acta. 1993.
DOI : 10.1002/hlca.19930760609.
Synthesis of 1,1-Bis(3,5-Dimethyl-2-Furyl)Ethene - the Chemo-Selectivity and Site-Selectivity of Its Cycloadditions
Heterocycles. 1993.
Regioselective and Stereoselective Thioamination of 7-Oxabicyclo[2.2.1]Hept-5-En-2-Yl Derivatives
Synlett. 1993.
1992
A Kinetically Stable Singlet-State of 1,2,4,5-Tetramethylenebenzene
Journal of the American Chemical Society. 1992.
Enantiomerically Pure 7-Oxabicyclo[2.2.1]Hept-5-En-2-Yl Derivatives (Naked Sugars) as Synthetic Intermediates .22. Stereoselective Synthesis of (1r)-1-C-(6-Amino-7h-Purin-8-Yl)-1,4-Anhydro-2,3-Dideoxy-3-Fluoro-D-Eryt Hro-Pentitol
Synlett. 1992.
Total Synthesis of Cyclophellitol Starting from Furan
Tetrahedron Letters. 1992.
DOI : 10.1016/S0040-4039(00)79144-1.
Total, Asymmetric-Synthesis of (1r)-1-C-(6'-Amino-7'h-Purin-8'-Yl)-1,4-Anhydro-3-Azido-2,3-Dideoxy-D-Er Ythro-Pentitol
Tetrahedron. 1992.
DOI : 10.1016/S0040-4020(01)88359-9.
Total Asymmetric-Synthesis of 3-Deoxy-Hexoses and 4-Deoxy-Hexoses and Derivatives
Tetrahedron. 1992.
DOI : 10.1016/S0040-4020(01)88356-3.
A Total, Asymmetric-Synthesis of 2-Deoxy-L-Fucose from Furan
Synthetic Communications. 1992.
Hetero-Diels-Alder Addition of Sulfur-Dioxide to 1,3-Dienes - Suprafaciality, Regioselectivity, and Stereoselectivity
Journal of the American Chemical Society. 1992.
DOI : 10.1021/ja00049a076.
Total Asymmetric Syntheses of D-Lividosamine and 2-Acetamido-2,3-Dideoxy-D-Arabino-Hexose Derivatives
Tetrahedron. 1992.
Should a Chemist Be Able to Do His Own Programming
Chimia. 1992.
Conformational-Analysis of Alpha-Methoxyketones - a Photoelectron Spectroscopic Investigation of 3-Methoxybicyclo[2.2.1]Heptan-2-Ones
Tetrahedron. 1992.
DOI : 10.1016/S0040-4020(01)88760-3.
The Diels-Alder Chemoselectivity of 3,4,6,7-Tetramethylidenebicyclo[3.2.1]Octane-2-Exo,8-Syn-Diyl Derivatives
Helvetica Chimica Acta. 1992.
DOI : 10.1002/hlca.19920750412.
Total Syntheses of 1,5-Dideoxy-1,5-Imino-D-Erythro-L-Allo-Octitol and (1s,2r,6r,7r,8s,8as)-Pentahydroxyindolizidine
Tetrahedron Letters. 1992.
Synthesis, Crystal-Structure and Reactivity of (Mu-3-Eta-2-7-Oxabicyclo[2.2.1]Hept-5-Yn-2-One)-Nonacarbonyldihydridotri Ruthenium and (Mu-3-Eta-2-7-Oxabicyclo[2.2.1]Hept-5-Yn-2-One)-Hexacarbonyldihydridotri S(Triphenylphosphine)Triruthenium
Bulletin De La Société Chimique De France. 1992.
Synthesis of Alpha-(1-]2)-, Alpha-(1-]3)-, Alpha-(1-]4)-, and Alpha-(1-]5)-C-Linked Disaccharides through 2,3,4,6-Tetra-O-Acetylglucopyranosyl Radical Additions to 3-Methylidene-7-Oxabicyclo[2.2.1]Heptan-2-One Derivatives
Journal of Organic Chemistry. 1992.
DOI : 10.1021/jo00033a032.
Substituent Effects on the Regioselectivity of the Baeyer-Villiger Oxidation of 7-Oxabicyclo[2.2.1]Heptan-2-Ones
Tetrahedron. 1992.
DOI : 10.1016/S0040-4020(01)88358-7.
1991
Asymmetric Total Synthesis of Azasugars Branched at C-5
Tetrahedron Letters. 1991.
Enantiomerically Pure 7-Oxabicyclo[2.2.1]Hept-5-En-2-Yl Derivatives (Naked Sugars) as Synthetic Intermediates .17. Total, Asymmetric-Synthesis of Hexoses and Azasugars Branched at C(5)
Tetrahedron. 1991.
DOI : 10.1016/S0040-4020(01)91030-0.
Enantiomerically Pure 7-Oxabicyclo[2.2.1]Hept-5-En-2-Yl Derivatives as Synthetic Intermediates .16. Total Asymmetric-Synthesis of 6-Deoxy-5-C-Methyl-D-Ribo-Hexose Structure in Aqueous-Solution
Carbohydrate Research. 1991.
DOI : 10.1016/0008-6215(91)89014-7.
Highly Stereoselective Synthesis of (+/-)-Aminobromocyclitol Derivatives from Furan
Synlett. 1991.
Total, Asymmetric-Synthesis of (+)-Castanospermine, (+)-6-Deoxycastanospermine, and (+)-6-Deoxy-6-Fluorocastanospermine
Journal of Organic Chemistry. 1991.
DOI : 10.1021/jo00006a031.
Radical Additions to Silyl Ketene Acetals - Introduction of C-Moieties to 7-Oxabicyclo[2.2.1]Hept-5-En-2-Endo-Ol
Tetrahedron Letters. 1991.
DOI : 10.1016/0040-4039(91)80814-M.
Enantiomerically Pure 7-Oxabicyclo[2.2.1]Hept-5-En-2-Yl Derivatives (Naked Sugar) as Synthetic Intermediates .15. a New Total Synthesis of D-Threo-L-Talo-Octose
Helvetica Chimica Acta. 1991.
DOI : 10.1002/hlca.19910740307.
Enantiomerically Pure 7-Oxabicyclo[2.2.1]Hept-5-En-2-Yl Derivatives (Naked Sugars) as Synthetic Intermediates .12. Highly Stereoselective Total Syntheses of Octoses and Derivatives
Journal of Organic Chemistry. 1991.
DOI : 10.1021/jo00003a041.
The Reactions of Gamma-Butyrolactone and Gamma-Butyrolactonol Derivatives, and of Tetrahydrofuran with Mixtures of Alcohols and Thionyl Chloride
Synlett. 1991.
Reaction of Dodecacarbonyltriruthenium with 7-Oxabicyclo[2.2.1]Hept-5-En-2-Yl Derivatives - Synthesis of (Mu-3-Eta-2-Benzyne)-Nonacarbonyldihydridotriruthenium and Derivatives
Journal of the Chemical Society, Chemical Communications. 1991.
Synthesis of Alpha-(1-]3)-Linked and Alpha-(1-]4)-Linked C-Disaccharides Using (+)-7-Oxabicyclo[2.2.1]Hept-5-En-2-One (Naked Sugar)
Tetrahedron Letters. 1991.
Substituent Effects on the Regioselectivity of One-Carbon Ring Expansions of 7-Oxabicyclo[2.2.1]Heptan-2-One Derivatives with Diazomethane
Tetrahedron Letters. 1991.
DOI : 10.1016/S0040-4039(00)74292-4.
Condensation of 2,3-Di(Methylidene)-7-Oxabicyclo[2.2.1]Heptane Derivatives into Dicarbonyl[Eta-3-Eta-3-Octa-2,6-Diene-1,8-Diyl]Iron Complexes with Nonacarbonyldiiron - Crystal-Structure of (1rs,2rs,3rs,4sr,5rs,6sr,1'rs,2'rs,3'rs,4'sr,5'rs,6'sr)-Dicarbonyl-((2,3 ,C-Eta-2',3',C-Eta)-2,2'-Ethylene-5,5',6,6'-Tetrakis[(Methanesulfonyloxy )-Methyl]-3,3'-Di(Methylidene)-Bis[7-Oxabicyclo[2.2.1]Hept-2-Yl)Iron
Helvetica Chimica Acta. 1991.
DOI : 10.1002/hlca.19910740418.
Highly Stereoselective Aminohydroxylations of Exo-2-Cyano-7-Oxabicyclo[2.2.1]Hept-5-En-2-Yl Acetate
Synthesis-Stuttgart. 1991.
1990
Optically Pure 7-Oxabicyclo[2.2.1]Hept-5-En-2-Yl Derivatives (Naked Sugars) as New Chirons
Synlett. 1990.
Synthesis of Rare Carbohydrates and Biomolecules from Furan
Bulletin Des Societes Chimiques Belges. 1990.
Application of New Optically Pure Ketene Equivalents Derived from Tartaric-Acids to the Total, Asymmetric Syntheses of (+)-6-Deoxycastanospermine and (+)-6-Deoxy-6-Fluorocastanospermine
Journal of the Chemical Society, Chemical Communications. 1990.
Stereoselective Syntheses of Protected Amino-Hydroxy-Cyclopentane-Carbaldehyde Derivatives from 7-Oxabicyclo[2.2.1]Hept-5-En-2-Yl Systems
Chimia. 1990.
New Chiral Auxiliaries and New Optically Pure Ketene Equivalents Derived from Tartaric-Acids - Improved Synthesis of (-)-7-Oxabicyclo[2.2.1]Hept-5-En-2-One
Tetrahedron-Asymmetry. 1990.
Enantiomerically Pure 7-Oxabicyclo[2.2.1]Hept-5-En-2-Yl Derivatives (Naked Sugars) as Synthetic Intermediates .11. Total Syntheses of (-)-Conduritol-B ((-)-1l-Cyclohex-5-Ene-1,3/2,4-Tetrol) and of (+)-Conduritol-F ((+)-1d-Cyclohex-5-Ene-1,2,4/3-Tetrol) - Determination of the Absolute-Configuration of (+)-Leucanthemitol
Helvetica Chimica Acta. 1990.
Total Synthesis of Branched-Chain Higher-Carbon Sugars - 1st Synthesis of Caldose, Calditol and 4-Deoxycalditol Stereoisomers
Tetrahedron Letters. 1990.
DOI : 10.1016/S0040-4039(00)88862-0.
Highly Stereoselective Total Syntheses of 2,5-Anhydro-3-Deoxy-D-Hexonic and 2,5-Anhydro-4-Deoxy-D-Hexonic Acids and of the Related Deoxyadenosines-C
Journal of Organic Chemistry. 1990.
DOI : 10.1021/jo00295a039.
Diels-Alder Additions of 1,3-Dienes to Propargylic Alcohols Catalyzed by the Wilkinsons Catalyst
Journal of Molecular Catalysis. 1990.
DOI : 10.1016/0304-5102(90)85067-R.
Synthesis of (1rs,2rs,5sr)-3,4,6,7-Tetramethylidene-8-Oxobicyclo[3.2.1]Oct-2-Yl Acetate and the Chemoselective and Stereoselective Coordination of Its Butadiene Functions with Rhodium and Iron Moieties
Organometallics. 1990.
DOI : 10.1021/om00160a028.
Through-Bond Interactions of Beta-Carbonyl and Beta-Imine Lone Pairs with Cationic 2p Orbital - Quantum Calculations on Bicyclo[2.2.2]Oct-1-Yl Cation and Derivatives
Journal of Organic Chemistry. 1990.
DOI : 10.1021/jo00309a012.
Synthesis and Circular-Dichroism of Optically Pure (+/-)-(1s,2s,5s)-5-Methoxy-3,4,6,7-Tetramethylidenebicyclo[3.2.1]Oct-2-Y L Derivatives - Bakers-Yeast Reduction of 4-Methoxy-5,6,7,8-Tetramethylidenebicyclo[2.2.2]Octan-2-One
Helvetica Chimica Acta. 1990.
DOI : 10.1002/hlca.19900730425.
Total, Asymmetric-Synthesis of Deoxypolyoxin-C
Tetrahedron. 1990.
DOI : 10.1016/S0040-4020(01)87887-X.
Regioselectivity of 7-Oxabicyclo[2.2.1]Hepta-2,5-Diene-Phenol Rearrangement as a Function of the Acid Promoter - Stereoselective Synthesis of 1,2,3,4-Tetrahydro-2-Hydroxynaphthalen-2-Yl Methyl Ketones
Tetrahedron Letters. 1990.
DOI : 10.1016/S0040-4039(00)94341-7.
Acid-Promoted Rearrangements of N-Substituted 8-Oxa-3-Azatricyclo[3.2.1.0/2,4]Octane-6,7-Dicarboxylates - Remote Substituent Effects on the Regioselectivity of the N-Acylaziridine/Dihydrooxazone Rearrangement
Helvetica Chimica Acta. 1990.
DOI : 10.1002/hlca.19900730316.
1989
The Stereoselective Methylations and Hydroxymethylations of 2,8-Dioxabicyclo[3.2.1]Octan-3-One Derivatives - Synthesis of Branched-Chain Sugars
Journal of the Chemical Society, Chemical Communications. 1989.
Polynuclear Iron and Rhodium Complexes of 7-Oxa[2.2.1]Hericene (2,3,5,6-Tetramethylidenebicyclo[2.2.1]Heptan-7-One)
Helvetica Chimica Acta. 1989.
DOI : 10.1002/hlca.19890720121.
A Highly Stereoselective Total Synthesis of (+/-)Castanospermine
Tetrahedron Letters. 1989.
DOI : 10.1016/S0040-4039(01)80287-2.
Enantiomerically Pure 7-Oxabicyclo[2.2.1]Hept-5-En-2-Yl Derivatives (Naked Sugars) as Synthetic Intermediates .7. Acid-Catalyzed Rearrangement of 3-Aza-8-Oxatricyclo[3.2.1.0/2,4]Octan-6-One Acetals - Highly Stereoselective Total Synthesis of 3-Amino-3-Deoxy-D-Altrose and Derivatives
Helvetica Chimica Acta. 1989.
DOI : 10.1002/hlca.19890720504.
Synthesis of (-)-Conduritol C (1l-Cyclohex-5-Ene-1,2,3/4-Tetrol)
Helvetica Chimica Acta. 1989.
Synthesis of Higher-Carbon Sugars Via Cross-Aldolization of 7-Oxanorbornan-2-One and Carbohydrate Aldehyde Derivatives
Journal of the Chemical Society, Chemical Communications. 1989.
Highly Stereoselective Total Syntheses of 2,5-Anhydro-4-Deoxy-D-Ribo-Hexonic Acid and of (1s)-1-C-(6-Amino-7h-Purin-8-Yl)-1,4-Anhydro-3-Deoxy-D-Erythro-Pentitol (= Cordycepin C)
Helvetica Chimica Acta. 1989.
DOI : 10.1002/hlca.19890720211.
The Electron-Releasing Homoconjugated Carbonyl Group - Application to the Total Syntheses of 3-Deoxy-, 4-Deoxy-Hexose, Lividosamine and Derivatives
Tetrahedron Letters. 1989.
DOI : 10.1016/S0040-4039(00)70712-X.
The Carbonyl Group as Homoconjugated Electron-Releasing Substituent - Regioselective Electrophilic Additions at Bicyclo[2.2.1]Hept-5-En-2-One, Bicyclo[2.2.2]Oct-5-En-2-One and Derivatives
Helvetica Chimica Acta. 1989.
DOI : 10.1002/hlca.19890720519.
Cyclo-Dimerization of 1-(Dimethoxymethyl)-5,6-Dimethylidene-7-Oxa-Bicyclo[2.2.1]Hept-2-Ene Induced by Nonacarbonyldiiron - Crystal-Structure of (1rs,2sr,3rs,4rs,4ars,9asr)-Tricarbonyl[C,2,3,C-Eta-(1,4-Epoxy-1,5-Bis(D Imethoxymethyl)-2,3-Dimethylidene-1,2,3,4,4a,9,9a,10-Octahydroanthracene )Iron)
Helvetica Chimica Acta. 1989.
Enantiomerically Pure 7-Oxabicyclo[2.2.1]Hept-5-En-2-Yl Derivatives (Naked Sugars) as Synthetic Intermediates .8. Total Synthesis of 2-(Beta-D-Ribofuranosyl)Thiazole-4-Carboxamide (Tiazofurin) and of Precursors of Ribo-C-Nucleosides
Helvetica Chimica Acta. 1989.
DOI : 10.1002/hlca.19890720819.
Total Synthesis of L-Allose, L-Talose, and Derivatives
Helvetica Chimica Acta. 1989.
DOI : 10.1002/hlca.19890720212.
Total Synthesis of Allonojirimycin (5-Amino-5-Deoxy-D-Allopyranose)
Angewandte Chemie, International Edition. 1989.
1988
Interaction between Non-Conjugated Chromophores .29. Circular-Dichroism of Planar, Exocyclic S-Cis-Butadienes Remotely Perturbed
Helvetica Chimica Acta. 1988.
DOI : 10.1002/hlca.19880710215.
Enantiomerically Pure 7-Oxabicyclo[2.2.1]Hept-5-En-2-Yl Derivatives as Synthetic Intermediates .3. Total Synthesis of D-Ribose and L-Ribose Derivatives
Helvetica Chimica Acta. 1988.
DOI : 10.1002/hlca.19880710316.
Syntheses and Tandem Diels-Alder Reactivities of 7,7-Diphenyl-[2.2.1]Hericene (= 7-(Diphenylmethylidene)-2,3,5,6-Tetramethylidenebicyclo[2.2.1]Heptane) and 7-Oxal[2.2.1]Hericene (= 2,3,5,6-Tetramethylidenebicyclo[2.2.1]Heptan-7-One)
Helvetica Chimica Acta. 1988.
DOI : 10.1002/hlca.19880710538.
Stereoselective Amino-Hydroxylation of the Double-Bond in 7-Oxabicyclo[2.2.1]Hept-5-En-2-Yl Derivatives - Remote Substituent Participation in Acid-Catalyzed Decompositions of Aziridines and Triazolines
Tetrahedron Letters. 1988.
DOI : 10.1016/S0040-4039(00)82156-5.
Synthesis and Circular-Dichroism of 5-Halogenobicyclo[2.2.1]Hept-5-En-2-Ones and 6-Halogenobicyclo[2.2.1]Hept-5-En-2-Ones - Tests for the Dekkers Quantitative Chirality Rule
Chimia. 1988.
Synthesis of (+)-1,3-2,5-Dianhydroviburnitol ((+)-(1r,2r,3s,5r,6s)-4,7-Dioxatricyclo[3.2.1.0/3,6]Octan-2-Ol)
Helvetica Chimica Acta. 1988.
Tandem Diels-Alder Reactivity Controlled by Remote Substituents - Regioselective Synthesis of Linearly Annellated 6-Membered Ring-Systems from (1rs,5sr,6rs,7sr)-6,7-Bis(Chloromethyl)-8,9-Dimethylidene-2-Oxabicyclo[3 .2.2]Nonan-3-One - Crystal-Structure of (1rs,5rs,6sr,11rs)-6,7-Bis(Chloromethyl)-3-Oxo-2-Oxatricyclo[7.4.0.0/1,5 ]Tridec-8-En-11-Yl Methyl Ketone
Helvetica Chimica Acta. 1988.
DOI : 10.1002/hlca.19880710537.
Abinitio Mo Calculations on the Rearrangements of 7-Oxa-2-Bicyclo[2.2.1]Heptyl Cations - the Facile Migration of Acyl Group in Wagner-Meerwein Rearrangements
Journal of Physical Organic Chemistry. 1988.
DOI : 10.1002/poc.610010507.
Synthesis of Optically Pure Tricarbonyliron Complexes of 5,6-Dimethylidenebicyclo[222]Oct-2-Yl Derivatives - Crystal-Structure and Absolute-Configuration of (+)-Tricarbonyl[(1s,2s,4r,5r,6s)-C,5,6,C-Eta-(5,6-Dimethylidenebicyclo[2 22]Oct-2-Yl P-Bromobenzoate)]Iron
Helvetica Chimica Acta. 1988.
DOI : 10.1002/hlca.19880710546.
Tandem Cheletropic Additions of Sulfur-Dioxide to [2.2.2]Hericene - the Barrelene Effect
Helvetica Chimica Acta. 1988.
DOI : 10.1002/hlca.19880710611.
The Reaction of Water with Iron Carbonyl and Ruthenium Carbonyl Complexes of Polyolefins - 1,2-Hydrogenation and 1,4-Hydrogenation of 1,3-Dienes - Hydrogenolysis of Allylic Ethereal Bonds and Deoxygenation of 7-Oxabicyclo[2.2.1]Hept-2-Enes
Helvetica Chimica Acta. 1988.
DOI : 10.1002/hlca.19880710547.
1987
Synthesis and Formation of Ironcarbonyl Complexes of 3',3'-Dimethyl-2,3,5,6-tetramethylidenespiro[bicyclo[2.2.1]heptane-7,2'-oxirane]. Single-Crystal and Molecular Structure of syn,exo2,3-anti,endo5,6-trans-m-[(1R,2R,3S,4S,5S,6R)-C,2,3,C-h:C,5,6,C-h-(3',3'-Dimethyl-2,3,5,6-tetra-methylidenespiro[bicyclo[2.2.1]heptane-7,2'-oxirane])]bis(tricarbonyliron)
Helvetica Chimica Acta. 1987.
DOI : 10.1002/hlca.19870700621.
Control of Diels-Alder Addition, Stereoselectivity and Regioselectivity by Remote Substituents and Tricarbonyl(Diene)Iron Moieties
Helvetica Chimica Acta. 1987.
Remote Tricarbonyl(Diene)Iron Substituent Effect on Ester Heterolysis - the Solvolyses of 5,6,7,8-Tetramethylidenebicyclo[2.2.2]Oct-2-Yl Methanesulfonate and of Its Tricarbonyliron Mononuclear and Dinuclear Complexes
Helvetica Chimica Acta. 1987.
Dynamic Modeling of Chemical-Reactions - the Diels-Alder Cycloaddition
Journal of Molecular Graphics. 1987.
Syntheses of (+)- and (-)-Methyl 8-Epinonactate and (+)- and (-)-Methyl Nonactate
Helvetica Chimica Acta. 1987.
DOI : 10.1002/hlca.19870700319.
Dynamic Modeling of Diels-Alder Reaction Using Computer-Graphics
Journal De Chimie Physique Et De Physico-Chimie Biologique. 1987.
Facile Migration of Acyl-Groups in Wagner-Meerwein Transpositions - Acid-Catalyzed Rearrangements of 5,6-Exo-Epoxy-7-Oxa-2-Bicyclo[2.2.1]Heptanone
Tetrahedron Letters. 1987.
Acid-Catalyzed Rearrangements of 5,6-Exo-Epoxy-7-Oxabicyclo(2.2.1)Hept-2-Yl Derivatives - Migratory Aptitudes of Acyl Vs Alkyl-Groups in Wagner-Meerwein Transpositions
Helvetica Chimica Acta. 1987.
Intramolecular Diels-Alder Reactions of 3h-Pyrroles Resulting from the Thermal Rearrangements of 2h-Pyrroles
Journal of Organic Chemistry. 1987.
DOI : 10.1021/jo00234a009.
Synthesis of Polyfunctional, Linearly Condensed 6-Membered Ring-Systems by Regioselective Tandem Diels-Alder Additions - Synthesis and Reactivity of 6,7-Bis(Chloromethyl)-8,9-Bis(Methylene)-2-Oxabicyclo[3.2.1]Nonan-3-One
Tetrahedron Letters. 1987.
DOI : 10.1016/S0040-4039(00)96090-8.
Interactions between Nonconjugated Chromophores .28. Regioselective Electrophilic Additions of Bicyclo[2.2.N]Alk-2-Enes Controlled by Remote Epoxide Functions
Helvetica Chimica Acta. 1987.
DOI : 10.1002/hlca.19870700723.
Interactions between Oxygen Lone-Pair Orbitals and Double-Bond Pi-Orbitals in Beta,Gamma-Unsaturated, Bicyclic Ketones - a Pe-Spectroscopic Investigation
Helvetica Chimica Acta. 1987.
DOI : 10.1002/hlca.19870700612.
Synthesis and Tandem Diels-Alder Reactivity of 1,3-Dimethoxy-5,6,7,8-Tetramethylidenebicyclo[2.2.2]Oct-2-Ene
Chimia. 1987.
Ironcarbonyl Complexes of 5,6-Dimethylidene-7-Oxabicyclo[2.2.1]Hept-2-Ene Derivatives - Synthesis of Substituted Tricarbonyl(Ortho-Quinodimethane)Iron Complexes and 2-Indanones
Helvetica Chimica Acta. 1987.
DOI : 10.1002/hlca.19870700715.
1986
Expeditious Syntheses of Methyl 8-Epi-Nonactate and Methyl Nonactate
Tetrahedron Letters. 1986.
DOI : 10.1016/S0040-4039(00)85280-6.
Naked Sugars as Synthetic Intermediates - Total Synthesis of L-Daunosamine
Journal of Organic Chemistry. 1986.
DOI : 10.1021/jo00376a055.
Regioselectivity of 1,3-Dipolar Cycloadditions Controlled by Remote Substitution and Lewis Acid Catalysts
Heterocycles. 1986.
Stereoselective Double Friedel-Crafts Acylation of Trans-Mu-(2,3,6,7-Tetramethylidenebicyclo[3.2.1]Octane)Bis(Tricarbonylir on) - Crystal-Structure of Trans-Mu-((1rs,2rs,3sr,5rs,6sr,7sr)-C,2,3,C-Eta-C,6,7,C-Eta-[(Z,Z)-1,1'- (3,7-Dimethylidenebicyclo[3.2.1]Octane-2,6-Diylidene)Di(2-Propanone)])Bi S(Tricarbonyliron)C
Helvetica Chimica Acta. 1986.
Interaction between Nonconjugated Chromophores .25. Diels-Alder Regioselectivity Controlled by Remote Substituents - the Cycloadditions of 1-(Dimethoxymethyl)-2,3-Dimethylidene-7-Oxabicyclo[2.2.1]Heptanes and 1-(Dimethoxymethyl)-2,3,5,6-Tetramethylidene-7-Oxabicyclo[2.2.1]Heptanes
Helvetica Chimica Acta. 1986.
Structure of (Alkene)Tetracarbonyliron Complexes - Variable-Temperature Circular-Dichroism of (5-Substituted 7-Oxabicyclo[2.2.1]Hept-2-Ene)Tetracarbonyliron Complexes
Organometallics. 1986.
DOI : 10.1021/om00143a016.
Experimental and Theoretical-Studies on the Homoconjugation in Bicyclic Carbenium and Oxonium Ions in the Gas-Phase
Tetrahedron Letters. 1986.
DOI : 10.1016/S0040-4039(00)83933-7.
Circular-Dichroism of Tricarbonyl(Diene)Iron Complexes - the Octant Rule Applied to Ketones Perturbed by Remote Fe(Co)3 Groups Crystal-Structure of (+/-Tricarbonyl[(1rs,4rs,5rs,6sr)-C,5,6,C-Eta-(5,6,7,8-Tetramethylidene- 2-Bicyclo[2.2.2]Octanone)]Iron
Helvetica Chimica Acta. 1986.
Synthesis and Diels-Alder Reactivity of 2,3,6,7-Tetrakis(Methylene)Bicyclo[3.2.1]Octane
Journal of Organic Chemistry. 1986.
DOI : 10.1021/jo00362a043.
Structure of Tricarbonyl(Diene)Iron Complexes in Solution - Variable-Temperature Circular-Dichroism of Trans-Mu-(2,3,5,6-Tetramethylidenebicyclo[2.2.2]Octane)Bis(Tricarbonylir on) Complexes
Helvetica Chimica Acta. 1986.
Long-Range Substituent Effects - the Regioselective Electrophilic Additions of Exo-3,6-Epoxytetrahydrophthalide and Its Derivatives
Tetrahedron Letters. 1986.
DOI : 10.1016/S0040-4039(00)85251-X.
Pyrimidalization of the Carbon-Atom of the Nitrogen-Carbon Double-Bond of 2-Azabicyclo[2.2.1]Hept-2-Enes - Radiocrystallographic Study and Calculations of Quantum-Mechanics
Nouveau Journal de Chimie. 1986.
Interaction between Nonconjugated Chromophores .26. Control of the Diels-Alder-Addition Regioselectivity by Remote Olefins - Syntheses and Cycloadditions of 2,3,5-Trimethylidenebicyclo[2.2.1]Heptane and 2,3,5,6,7-Pentamethylidenebicyclo[2.2.2]Octane
Helvetica Chimica Acta. 1986.
DOI : 10.1002/hlca.19860690604.
Regioselectivity of Electrophilic Additions to 7-Oxabicyclo[2.2.1]Heptenes Controlled by Remote Substituents - Arenesulfonyl Substituted 7-Oxabicyclo[2.2.1]Heptenes as Stereoselective and Regioselective Chiral Dienophiles
Journal of Organic Chemistry. 1986.
DOI : 10.1021/jo00376a054.
Conformational-Analysis of Endoperoxides Grafted onto Bicyclo[2.2.N]Alkanes as a Test of the Rigidity of the Bicyclic Skeleton - Photooxidation of [2.2.2]Hericene and 2,3,5,6-Tetramethylidenebicyclo[2.2.N]Alkanes .24
Helvetica Chimica Acta. 1986.
DOI : 10.1002/hlca.19860690403.
Chemoselective and Stereoselective Functionalization of 7-Oxabicyclo[2.2.1]Hept-5-En-2-One with Dichloroketene
Tetrahedron Letters. 1986.
DOI : 10.1016/S0040-4039(00)85250-8.
1985
Stereoselective Nucleophilic Additions to a Bicyclic Ketone Controlled by a Remote Tricarbonyl(Diene)Iron Moiety
Angewandte Chemie, International Edition. 1985.
Electrophilic Additions Controlled by Remote Substituents - Total Synthesis of Daunosamine
Tetrahedron Letters. 1985.
DOI : 10.1016/S0040-4039(00)98879-8.
Interaction between Non-Conjugated Chromophores .23. 233 Face Selectivity of the Diels-Alder Additions of Sulfur-Substituted Dienes and Tetraenes Grafted onto 7-Oxabicyclo[2.2.1]Heptanes
Helvetica Chimica Acta. 1985.
The Synthesis of (+/-)-11-Deoxydaunomycinone Via Regioselective Tandem Diels-Alder Reactions
Helvetica Chimica Acta. 1985.
Face Selectivity of the Diels-Alder Reaction of Hexadienone Moieties Grafted onto the Bicyclo[2.2.2]Octene Skeleton and Perturbed by a Remote Tricarbonylbutadieneiron Group
Helvetica Chimica Acta. 1985.
DOI : 10.1002/hlca.19850680529.
Stereoselective Double Functionalization of Iron-Carbonyl Complexes of 5,6,7,8-Tetramethylidenebicyclo[2.2.2]Oct-2-Ene - Crystal-Structure and Absolute-Configuration of (-)-Trans-Mu-[(2s,5r,7s)-C,5,6,C-Eta-C,7,8,C-Eta-(6,7,8-Trimethylidene-5 -((Z)-2-Oxopropylidene)-2-Bicyclo[2.2.2]Octyl Acetate)]-Bis(Tricarbonyliron)O
Helvetica Chimica Acta. 1985.
Experimental and Abinitio Molecular-Orbital Studies on Collisions of Ch4+. and Ch5+ with Molecular-Oxygen - on the Formation of Methane (Ch4(2+)) and Methonium (Ch5(2+)) Dications and Stable Chn-Species (N = 0-3)
Journal of the American Chemical Society. 1985.
Interaction between Non-Conjugated Chromophores .22. Synthesis and Diels-Alder Reactivity of 1-(Dimethoxy)Methyl-2,3,5,6-Tetramethylidene-7-Oxabicyclo[2.2.1]Heptane
Helvetica Chimica Acta. 1985.
H-1-Nmr Spectra of Cyclohexa-1,4-Dienes and Cyclohexenes Annellated to Bicyclo[2.2.1]Hept-2-Enes - the Inter-Ring Homoallylic H,H Coupling-Constants as Stereochemical Probes
Helvetica Chimica Acta. 1985.
DOI : 10.1002/hlca.19850680814.
2,3-Bis(Methylene)Bicyclo[2.1.1]Hexane and 3,4-Bis(Methylene)Tricyclo[3.1.0.02,6]Hexane - Interaction between a Pi-System and a Cyclobutane or Bicyclobutane Moiety
Journal of Organic Chemistry. 1985.
(2,3-Bis(Methylene)Bicyclo[2.2.2]Octane)Zirconocene - Synthesis, Structure, and Electrochemical Reduction
Z. Naturforsch. B. 1985.
Double-Bond Pyramidalization in Bicyclic Alkanes - Abinitio Mo Calculations on Bicyclo[2.2.1]Hept-2-Ene, Bicyclo[2.1.1]Hex-2-Ene and Bicyclo[3.2.1]Oct-6-Ene Derivatives
Journal of Molecular Structure: Theochem. 1985.
Face Selectivity in the Diels-Alder Additions and Chelotropic Addition of Sulfur-Dioxide to 2-(D)Methylidene-3-Methylidenebicyclo[2.2.1]Heptane
Helvetica Chimica Acta. 1985.
DOI : 10.1002/hlca.19850680628.
1984
Variable temperature circular dichroism of tricarbonyl(1,3-diene)iron complexes
Inorganica Chimica Acta. 1984.
DOI : 10.1016/S0020-1693(00)82524-4.
Stereoselective control in the base-catalyzed hydrogen/deuterium exchange of 5,6-dimethylidene-2-bicyclo[2.2.n]alkanone tricarbonyliron complexes. Revision of the structures of tricarbonyliron complexes of 5,6-dimethylidenebicyclo[2.2.2]oct-2-ene and 5,6-dimethylidenebicyclo[2.2.1]hept-2-ene
Helvetica Chimica Acta. 1984.
DOI : 10.1002/hlca.19840670410.
Monoolefin and diene cycloaddition induced by transition-metal carbonyls. Cyclodimerization of 5,6-dimethylidene-7-oxabicyclo[2.2.1]hept-2-ene catalyzed by dodecacarbonyltriosmium
Helvetica Chimica Acta. 1984.
DOI : 10.1002/hlca.19840670632.
The Circular-Dichroism of 5,6-Dimethylidene-2-Bicyclo[2.2.N]Alkyl Esters - Chiral Exciton Coupling between Benzoate and Exocyclic S-Cis-Butadiene Chromophores
Helvetica Chimica Acta. 1984.
DOI : 10.1002/hlca.19840670228.
2,5-Bis[[(Z)-(2-Nitrophenyl)Sulfenyl]Methylene]-3,6-Dimethylene-7-Oxabic Yclo[2.2.1]Heptane - a Versatile Reagent for Tandem Regioselective Diels-Alder Reactions
Journal of Organic Chemistry. 1984.
DOI : 10.1021/jo00187a046.
Macrocycles by Intramolecular Diels-Alder Reaction - Regioselective Synthesis of Anthracycline Precursors
Angewandte Chemie, International Edition. 1984.
A Doubly-Convergent and Regioselective Synthesis of (+/-)-Daunomycinone
Tetrahedron. 1984.
DOI : 10.1016/S0040-4020(01)91514-5.
The Non-Planarity of the Bicyclo[2.2.1]Hept-2-Ene Double-Bond - Crystal-Structures of Bicyclo[2.2.2]Oct-2-Ene, Bicyclo[2.2.1]Hept-2-Ene, and Bicyclo[2.1.1]Hex-2-Ene Systems
Helvetica Chimica Acta. 1984.
DOI : 10.1002/hlca.19840670428.
Diels-Alder Stereoselectivity and Regioselectivity Controlled by Remote Substituents and Solvent - Cyclo-Additions of 1-(Dimethoxymethyl)-2,3-Bis(Methylene)-7-Oxabicyclo[2.2.1]Heptane
Tetrahedron Letters. 1984.
Conformational-Analysis of 2,3,5,6-Tetrakis(Methylene)Bicyclo[2.2.2]Octanes by Circular-Dichroism
Tetrahedron Letters. 1984.
DOI : 10.1016/S0040-4039(01)81157-6.
The Carbonyl Group as Homoconjugated Electron Donating Substituent - Abinitio Sto 3g Mo Calculations
Tetrahedron Letters. 1984.
DOI : 10.1016/S0040-4039(01)81315-0.
Optical Resolution of 7-Oxabicyclo[2.2.1]Hept-2-Ene Derivatives - Diastereoselectivity in the Formation of Cyanohydrine-Brucine Complexes
Helvetica Chimica Acta. 1984.
DOI : 10.1002/hlca.19840670629.
1983
The Circular-Dichroism of 2,3-Dimethylidene-5-Norbornyl Derivatives
Tetrahedron Letters. 1983.
DOI : 10.1016/S0040-4039(00)88180-0.
Dynamic Representation of Quantum Chemical Results Using Computer-Graphics - Molecular-Rearrangements, Art or Science
Journal of Molecular Structure: Theochem. 1983.
The Preparation of Optically Pure 7-Oxabicyclo[2.2.1]Hept-2-Ene Derivatives - the Cd Spectrum of (+)-(1r)-7-Oxabicyclo[2.2.1]Hept-5-En-2-One
Helvetica Chimica Acta. 1983.
DOI : 10.1002/hlca.19830660627.
Control of the Diels-Alder Addition Regioselectivity by Remote Substituents - Synthesis of Anthracycline Precursors
Tetrahedron Letters. 1983.
DOI : 10.1016/S0040-4039(00)81691-3.
Interaction between Non-Conjugated Chromophores .19. Crystal and Molecular-Structure of 2,3,5,6,7,8-Hexamethylidenebicyclo[2.2.2]Octane ([2.2.2]Hericene)
Helvetica Chimica Acta. 1983.
DOI : 10.1002/hlca.19830660521.
Interaction between Non-Conjugated Chromophores .18. Preparation and Diels-Alder Reactivity of 2,3,5,6,7,8-Hexamethylidenebicyclo[2.2.2]Octane ([2.2.2]Hericene) - Force-Field Calculations of Exocyclic Dienes as a Moiety of Bicyclic Skeletons
Helvetica Chimica Acta. 1983.
DOI : 10.1002/hlca.19830660103.
Vapor-Phase Uv Spectra of 2,3,5,6,7,8-Hexakis(Methylene)Bicyclo [2.2.2] Octane ([2.2.2] Hericene) and Related S-Cis-Butadiene Derivatives
Canadian Journal of Spectroscopy. 1983.
Interactions between Homoconjugated Diene and Epoxide Functions - Effect on Diels-Alder Regioselectivity
Tetrahedron Letters. 1983.
DOI : 10.1016/S0040-4039(00)88179-4.
Site of Protonation and Conformational Effects on Gas-Phase Basicity in Beta-Amino Alcohols - the Nature of Internal H-Bonding in Beta-Hydroxy Ammonium-Ions
Journal of the American Chemical Society. 1983.
DOI : 10.1021/ja00349a006.
Preparation and Diels-Alder Reactivity of Tricarbonyliron Complexes of [2.2.2]Hericene
Helvetica Chimica Acta. 1983.
DOI : 10.1002/hlca.19830660729.
Stereoselective Control in the Base-Catalyzed H-D Exchange-Reaction of 5,6,7,8-Tetrakis(Methylene)-2-Bicyclo[2.2.2]Octanone Irontricarbonyl Complexes
Tetrahedron Letters. 1983.
DOI : 10.1016/S0040-4039(00)81822-5.
Interaction between Non-Conjugated Chromophores .20. Synthesis and Diels-Alder Reactivity of 5,6,7,8-Tetramethylidene-2-Bicyclo[2.2.2]Octanol and Octanone - Selective Oxidations of the Corresponding Bis (Irontricarbonyl) Complexes
Helvetica Chimica Acta. 1983.
DOI : 10.1002/hlca.19830660417.
Interaction between Non-Conjugated Chromophores .20. Face Selectivity of the Diels-Alder Reaction of 5,6-Bis((D)Methylidene)-2-Bicyclo[2.2.2]Octene
Helvetica Chimica Acta. 1983.
DOI : 10.1002/hlca.19830660427.
1982
Exocyclic Dienes and the Synthesis of Anthracyclins
Chimia. 1982.
Stereochemistry and Reactivity of Pi-Systems
Chimia. 1982.
Carbonyliron-Assisted Cycloaddition of a 1,3-Diene to a Cc Double-Bond - Synthesis of an Anthracyclinone Precursor
Angewandte Chemie, International Edition. 1982.
Copper(I)-Catalyzed and Copper(Ii)-Catalyzed Diels-Alder Additions of Alpha-Substituted Acrylonitrile to Furan - the Synthesis of "7-Oxa-Bicyclo[2.2.1]Hept-5-En-2-One
Helvetica Chimica Acta. 1982.
DOI : 10.1002/hlca.19820650604.
Face Selectivity of the Diels-Alder Additions of Exocyclic Dienes Grafted onto 7-Oxabicyclo[2.2.1]Heptanes
Helvetica Chimica Acta. 1982.
DOI : 10.1002/hlca.19820650321.
Interaction between Non-Conjugated Chromophores .17. Effects of Remote Substitution on the Photooxidation of Exocyclic S-Cis-Butadienes Grafted onto Bicyclo[2.2.1]Heptanes - Thermal and Rhodium Catalyzed Rearrangements of 3,6-Dihydro-1,2-Dioxines
Helvetica Chimica Acta. 1982.
DOI : 10.1002/hlca.19820650322.
Chemoselective, Regioselective, and Stereoselective Hydroalumination of 7,8-Epoxy-2,3,5,6-Tetramethylenebicyclo[2.2.2]Octane
Journal of Organic Chemistry. 1982.
DOI : 10.1021/jo00138a022.
(2,9-6,12-Eta-2,3,5,6-Tetrakis(Methylene)-Bicyclo[2.2.2]Octane)Zirconoce Ne, an Isolable Bis(Olefin)Zirconium(Ii) Compound
Angewandte Chemie, International Edition. 1982.
Synthesis and Diels-Alder Reactivity of 7-Isopropylidene-2,3,5,6-Tetramethylenebicyclo-[2.2.1]Heptane (7,7-Dimethyl[2.2.1]Hericene)
Journal of Organic Chemistry. 1982.
Regioselective Additions of Electrophiles to Olefins Remotely Perturbed - the Carbonyl Group as a Homoconjugated Electron Donating Substituent
Tetrahedron Letters. 1982.
DOI : 10.1016/S0040-4039(00)87396-7.
Interaction between Non-Conjugated Chromophores .15. Face Selectivity of the Diels-Alder Additions of 2-Substituted 5,6-Bis((E)-Chloromethylidene)Bicyclo[2.2.2]Octanes
Helvetica Chimica Acta. 1982.
Interactions between Non-Conjugated Chromophores .13. Interaction between Exocyclic S-Cis-Butadiene and Homoconjugated Functions - Preparation and Diels-Alder Reactivity of Remotely Substituted 2,3-Dimethylidenebicyclo[2.2.2]Octanes
Helvetica Chimica Acta. 1982.
Interaction between Non-Conjugated Chromophores .14. Regioselectivity of the Diels-Alder Additions of 2-Substituted 5,6-Dimethylidenenorbornanes and Dimethylidenebicyclo[2.2.2]Octanes
Helvetica Chimica Acta. 1982.
1981
Stereospecific functionalizations of iron carbonyl complexes of 5,6,7,8-tetrakis(methylene)bicyclo[2.2.2]oct-2-ene. Crystal and molecular structure of (C12H12)Fe2(CO)6
Journal of Organometallic Chemistry. 1981.
DOI : 10.1016/S0022-328X(00)86720-0.
Stereoselective acetylation of iron carbonyl complexes of 5,6,7,8-tetrakis(methylene)bicyclo[2.2.2]oct-2-ene. Diene-heterotriene tricarbonyliron coordination equilibrium in solution and crystal structure of (C12H11COCH3)Fe2(CO)6
Journal of Organometallic Chemistry. 1981.
DOI : 10.1016/S0022-328X(00)86721-2.
Regioselective addition of protic acids to tricarbonyliron complexes of 2,3,5,6-tetrakis(methylene)-7-oxabicyclo[2.2.1]heptane. Crystal structure of (C10H10O)Fe2(CO)6
Journal of Organometallic Chemistry. 1981.
DOI : 10.1016/S0022-328X(00)82287-1.
Inductive and polarizability effects of an exocyclic diene-iron tricarbonyl group. The acetolyses of exo- and endo-irontricarbonyl complexes of 5,6-dimethylidene-2-exo-norbornyl and 2,3-dimethylidene-7-anti-norbornyl parabromobenzenesulfonates
Helvetica Chimica Acta. 1981.
DOI : 10.1002/hlca.19810640846.
Crystal structure and absolute configuration of (+)-(1S,2R)-5,6-dimethylidene-2-exo-norbornyl-exo-irontricarbonyl p-bromobenzoate
Helvetica Chimica Acta. 1981.
DOI : 10.1002/hlca.19810640738.
New Dienophiles - 1-Acetylvinyl Arenecarboxylates - Reactivity toward Cyclopentadiene and Exocyclic Dienes
Helvetica Chimica Acta. 1981.
DOI : 10.1002/hlca.19810640121.
Non-Planarity of Pi-Systems in 5,6-Bis(Methylene)-7-Oxanorborn-2-Ene
Journal of the American Chemical Society. 1981.
DOI : 10.1021/ja00398a039.
Synthesis and Diels-Alder Reactivity of 2,3,5,6-Tetramethylidenenorbornane
Helvetica Chimica Acta. 1981.
DOI : 10.1002/hlca.19810640812.
The Pi-Anisotropy of the Double-Bond of a Syn-11-Oxasesquinorbornene Derivative-1) - Stereoselectivity of the Diels-Alder Additions of (2-Norborneno)[C]Furan2) - Crystal-Structure of 11-Oxa-Endo-Tetracyclo[6.2.1.13,6.02,7]-Dodec-2(7)-Ene-9,10-Exo-Dicarbox Ylic Anhydride
Helvetica Chimica Acta. 1981.
DOI : 10.1002/hlca.19810640613.
Thermoneutral Dyotropic Transfer of Hydrogen in a Hydrocarbon
Journal of the American Chemical Society. 1981.
DOI : 10.1021/ja00403a059.
Charge-Transfer Bands of Bicyclic Beta,Gamma-Unsaturated Ketones - Circular-Dichroism of (+)-(1r)-5,6-Dimethylidene-2-Bicyclo[2.2.2]Octanone and (+)-(1r)-2-Bicyclo[2.2.2]Oct-5-Enone
Tetrahedron Letters. 1981.
DOI : 10.1016/S0040-4039(01)83022-7.
Crystal-Structure and Absolute-Configuration of (+)-(1s,2r)-5,6-Dimethylidene-2exo-Norbornyl-Exo-Irontricarbonyl Para-Bromobenzoate
Helvetica Chimica Acta. 1981.
Acetolyses of Pi-Irontricarbonyl Complexes of 2,3-Dimethylidene-7anti-Norbornyl and 5,6-Dimethylidene-2exo-Norbornyl Esters
Tetrahedron Letters. 1981.
DOI : 10.1016/0040-4039(81)80063-9.
1980
Stereoselective oxidation of ruthenium and iron carbonyl complexes of 5,6,7,8-tetrakis(methylene)bicyclo[2.2.2]oct-2-ene
Journal of Organometallic Chemistry. 1980.
DOI : 10.1016/S0022-328X(00)90342-5.
Iron carbonyl complexes of 2,3,5,6-tetrakis(methylene)-7-oxabicyclo[2.2.1]heptane. Crystal and molecular structure of (C10H10O)Fe(CO)3 and (C9H10CO)Fe2(CO)6
Journal of Organometallic Chemistry. 1980.
DOI : 10.1016/S0022-328X(00)89872-1.
O-17 Nuclear Magnetic-Resonance - the Effects of Remote Unsaturation on O-17-Chemical Shifts in Polycyclic Ethers
Tetrahedron. 1980.
The Acetolysis of Exo-5,6-Dimethylidene-2-Norbornyl and Endo-5,6-Dimethylidene-2-Norbornyl Para-Bromobenzenesulfonates and of Their Optically-Active and Deuterium-Labeled Derivatives
Helvetica Chimica Acta. 1980.
Interaction between Non-Conjugated Chromophores .2. Optical-Activity in Remotely Perturbed Exocyclic S-Cis-Butadienes - Preparation and Circular-Dichroism of Enantiomerically Pure 5,6-Dimethylidene-2-Norbornyl Derivatives
Helvetica Chimica Acta. 1980.
Interactions between Non-Conjugated Chromopheres .12. the Photochemistry of 5,6-Dimethylidene-2-Norbornanone - Synthesis and Diels-Alder Reactivity of 2,3-Dimethylidenebicyclo-[2.1.1]Hexane
Helvetica Chimica Acta. 1980.
DOI : 10.1002/hlca.19800630508.
2,3,5,6,7,8-Hexakis(Methylene)Bicyclo[2.2.2]Octane
Angewandte Chemie, International Edition. 1980.
Radical Cation States of 2,3,5,6,7,8-Hexamethylidenebicyclo[2.2.2]Octane
Helvetica Chimica Acta. 1980.
DOI : 10.1002/hlca.19800630304.
An Efficient Synthesis of 2,3,5,6-Tetramethylidene-7-Oxanorbornane
Helvetica Chimica Acta. 1980.
DOI : 10.1002/hlca.19800630506.
Asymmetric Induction in the Rearrangement of Monocyclic Endoperoxides into Gamma-Hydroxy-Alpha-Beta-Unsaturated Aldehydes
Journal of the Chemical Society, Chemical Communications. 1980.
Interaction between Non-Conjugated Chromophores .10. 7,8-Epoxy-2,3,5,6-Tetrakis(Methylene)Bicyclo[2.2.2]Octane - Synthesis and Diels-Alder Reactivity
Tetrahedron. 1980.
DOI : 10.1016/0040-4020(80)85037-X.
The Homoallyl-Cyclopropylcarbinyl Cation Rearrangement in the Solvolyses of Exo-5-Norbornen-2-Yl and Endo-5-Norbornen-2-Yl Para-Bromobenzenesulfonates - Application of 2h-Nmr. Spectroscopy
Helvetica Chimica Acta. 1980.
Anthracyclinones .2. Synthesis of (+/-)-4-Demethoxydaunomycinone by Double Diels-Alder Additions to 2,3,5,6-Tetramethylidene-7-Oxanorbornane
Helvetica Chimica Acta. 1980.
Unambiguous Proof for Alcoxycarbonyl-Group Migration in Wagner-Meerwein Rearrangements
Helvetica Chimica Acta. 1980.
DOI : 10.1002/hlca.19800630849.
Stereoselectivity of the Diels-Alder Additions of Exocyclic Dienes Grafted onto Bicyclo[2.2.Normal]Alkanes
Tetrahedron Letters. 1980.
DOI : 10.1016/S0040-4039(00)77436-3.
1979
Iron, molybdenum and tungsten carbonyls of 5,6,7,8-tetrakis(methylene)bicyclo[2.2.2]oct-2-ene. Crystal and molecular structure of (C12H12)Fe(CO)3
Inorganica Chimica Acta. 1979.
DOI : 10.1016/S0020-1693(00)89387-1.
Iron and ruthenium carbonyls of 2,3,5,6-tetrakis(methylene)bicyclo[2.2.2]octane. Crystal and molecular structure of (C12H14)Fe(CO)3
Inorganica Chimica Acta. 1979.
DOI : 10.1016/S0020-1693(00)93439-X.
Iron and Ruthenium Carbonyls of 6,7-Dimethylene-Exo-3-Oxatricyclo[3.2.1.02,4]Octane - Protic Acid Additions to an Epoxide Ring Homoconjugated to a Eta-4-(Diene)Fe(Co)3 Function - Crystal-Structures of (C9h10o)Fe(Co)3 and (C10h14o2)Fe(Co)3
Journal of Organometallic Chemistry. 1979.
DOI : 10.1016/S0022-328X(00)96166-7.
Secondary 2-Norbornyl Cation Intermediates Substituted at C(5) and C(7) by Electron-Withdrawing Groups - Addition of Fluorosulfuric Acid to Unsaturated Norbornane Derivatives
Helvetica Chimica Acta. 1979.
DOI : 10.1002/hlca.19790620137.
Interaction between Non-Conjugated Chromophores .9. Effects of Homoconjugated Cyclopropane and Oxirane Rings on the Diels-Alder Reactivity of 2,3-Bis(Methylidene)Norbornane
Helvetica Chimica Acta. 1979.
DOI : 10.1002/hlca.19790620731.
Radical Cation States of 2,3,5,6-Tetramethylenenorbornane, 2,3,5,6-Tetramethylenebicyclo[2.2.2]Octane and of Related Compounds
Recueil des Travaux Chimiques des Pays-Bas. 1979.
Conformational-Analysis and the Rearrangements of (Norborn-2-Eno)[D](3,6-Dihydro-1,2-Dioxine)
Tetrahedron Letters. 1979.
Conference Papers
2009
Phosphineless iron-catalyzed carbon-carbon bond cross-coupling reactions
2009. p. 229-ORGN.
New organic chemistry of sulfur dioxide: Asymmetric total synthesis of polypropionate antibiotics
2009. p. 454-ORGN.
Depletion of the intracellular coenzyme NAD plus in activated T-cells ameliorates experimental autoimmune encephalomyelitis
2009. 25th Congress of the European-Committee-for-Treatment-and-Research-in-Multiple-Sclerosis , Dusseldorf, GERMANY , Sep 09-12, 2009. p. S178-S178.
2008
Use of sultines in the asymmetric synthesis of polypropionate antibiotics
2008. 21st International Congress for Heterocyclic Chemistry , Sydney, AUSTRALIA , Jul 15-20, 2007. p. 791-805.
DOI : 10.1351/pac200880040791.
2007
Conduramine F-1 epoxides: synthesis and their glycosidase inhibitory activities
2007. 8th Tetrahedron Symposium on Challenges in Organic Chemistry , Berlin, GERMANY , Jun 27-29, 2007. p. 6558-6572.
DOI : 10.1016/j.tet.2007.03.149.
2004
C-linked disaccharides analogues of the T epitope: Toward an artificial anti-cancer vaccine
2004. p. U224-U224.
2003
One-pot three- and four-component synthesis of polyfunctional sulfones, sulfonic esters, and sulfonamides
2003. p. U162-U162.
1995
Asymmetric Syntheses of Herbicidine Undecoses and of C-Galactosides of Cyclitols Starting with Furan
1995. p. 38-CARB.
1989
The Electron-Donating Carbonyl Group Total Synthesis of Rare Sugars
1989. p. 114-ORGN.
Total Synthesis of Castanospermine and Other Potential Glycosidase Inhibitors
1989. p. 23-CARB.
1988
Total Synthesis of Aminodeoxyhexoses Via the Amino-Hydroxylation of 7-Oxanorbornene Derivatives
1988. p. 72-ORGN.
Tandem Cheletropic Additions of So2 to [2.2.2]Hericene - the Barrelene Effect
1988. p. 23-ORGN.
Synthesis of Rare Carbohydrates from 7-Oxanorbornenes (Naked Sugars)
1988. p. 292-ORGN.
1987
Synthesis of Carbohydrates and Derivatives from 7-Oxanorbornenes (Naked Sugars)
1987. p. 35-CARB.
Synthesis of Polyfunctional, Linearly Condensed 6-Membered Ring-Systems by Regioselective Tandem Diels-Alder Additions
1987. p. 151-ORGN.
1986
Total Asymmetric Syntheses of Conduritol-C and Conduritol-D, and of a Cyanoglucoside
1986. p. 14-ORGN.
1985
Naked Sugars as Synthetic Intermediates - Stereospecific Synthesis of L-Daunosamine
1985. p. 62-ORN.
Face Selectivity in the Diels-Alder Additions and Chelotropic Reaction of Sulfur-Dioxide of 2-Deuteriomethylene-3-Methylenebicyclo[2.2.1]Heptane
1985. p. 40-ORN.
Reviews
2009
Desulfinylation of Prop-2-enesulfinic Acid: Experimental Results and Mechanistic Theoretical Analysis
Journal Of The American Chemical Society. 2009.
DOI : 10.1021/ja901565a.
2008
Combinatorial synthesis of linearly condensed polycyclic compounds, including anthracyclinones, through tandem Diels-Alder additions
Anthracycline Chemistry And Biology I: Biological Occurence And Biosynthesis, Synthesis And Chemistry. 2008.
DOI : 10.1007/128_2007_148.
Theses
2011
Synthesis of C-linked Disaccharides and Analogues as Biomimetics of the TF Epitope
Lausanne, EPFL, 2011.
DOI : 10.5075/epfl-thesis-4808.
2010
Total Synthesis of Dolabriferol and Polypropionate Fragments Applying New Organic Chemistry of Sulfur Dioxide
Lausanne, EPFL, 2010.
DOI : 10.5075/epfl-thesis-4788.
Synthesis of Glycomimetics as Potential Anti-Cancer Agents
Lausanne, EPFL, 2010.
DOI : 10.5075/epfl-thesis-4764.
Dissymmetrical Double-Chain Elongation Approach to the Asymmetric Synthesis of Long-Chain Polypropionates
Lausanne, EPFL, 2010.
DOI : 10.5075/epfl-thesis-4756.
Access to long-chain polyketides by double-elongation reactions
Lausanne, EPFL, 2010.
DOI : 10.5075/epfl-thesis-4608.
2009
New developments in iron-catalyzed carbon-carbon bond forming reactions
Lausanne, EPFL, 2009.
DOI : 10.5075/epfl-thesis-4517.
Search for new anti-cancer heterocyclic compounds
Lausanne, EPFL, 2009.
DOI : 10.5075/epfl-thesis-4444.
New efficient synthetic strategies towards the AB and CD spiroketal fragments of spongistatins and analogues
Lausanne, EPFL, 2009.
DOI : 10.5075/epfl-thesis-4383.
2007
New efficient synthetic routes toward functionalised polyketides
Lausanne, EPFL, 2007.
DOI : 10.5075/epfl-thesis-3800.
Development of new anticancer agents based on [alpha]-mannosidase inhibition
Lausanne, EPFL, 2007.
DOI : 10.5075/epfl-thesis-3793.
Book Chapters
2009
Anomeric effects in pyranosides and related acetals
Carbohydrate Chemistry. Chemical and Biological Approaches; RCS Publishing, 2009. p. 13-32.
2007
Imino-C-disaccharides and analogues: synthesis and biological activity
Iminosugars: from synthesis to therapeutic applications; Wiley, 2007. p. 87-131.
2006
Trifluoromethanesulfonyl chloride, first update
Electronic Encyclopedia of Reagents for Organic Synthesis; 2006.
1996
A New and Practical Removal of Allyl and Allyloxycarbonyl Groups Promoted by Water-Soluble Pd(0) Catalysts
The Roots of Organic Development; Amsterdam: Elsevier, 1996. p. 416-430.
1989
Synthesis of Carbohydrates and Derivatives from 7-Oxanorbornenes (Naked Sugars)
Acs Symposium Series; 1989. p. 197-241.
Patents
2010
Novel dihydroxypyrrolidine derivatives as anti-cancer agents
2010.
WO2009118712
2009
Derivatives of dihydroxypyrrolidine as anti- cancer compounds
2009.
WO2009072062
EP2067771
2004
Polyfunctional sulfonamides and sulfonates and process for preparing them
2004.
1994
DEALLYLATION REAGENT AND DEALLYLATION METHOD USING SAID REAGENT
1994.
ES2166372
AT211725
EP0693052
HU218397
US5773617
HUT76715
EP0693052
NO953976
FI954765
FR2703688
WO9424088
CA2160163
FR2703688
Catalytic process useful for selectively cleaving a protected functional group and molecules capable of being deprotected according to this process
1994.
FR2703687