Complete Publication List

Journal Articles

2019

Alkynylation of radicals: spotlight on the “Third Way” to transfer triple bonds

F. Le Vaillant; J. Waser 

Chemical Science

2019-10-21

Vol. 10 , num. 39, p. 8909-8923.

DOI : 10.1039/c9sc03033f

1,3-Difunctionalization of Aminocyclopropanes via Dielectrophilic Intermediates

M-M. Wang; J. Waser 

Angewandte Chemie-International Edition

2019-09-23

Vol. 58 , num. 39, p. 13880-13884.

DOI : 10.1002/anie.201907060

An Alternative One-Electron Oxidation Strategy to Access Hypervalent Iodine Reagents

J. Ceballos; M. Garreau; J. Waser 

Chem

2019-09-12

Vol. 5 , num. 9, p. 2287-2289.

DOI : 10.1016/j.chempr.2019.08.005

Palladium-Catalyzed Carboxy-Alkynylation of Propargylic Amines Using Carbonate Salts as Carbon Dioxide Source

P. D. G. Greenwood; J. Waser 

European Journal Of Organic Chemistry

2019-09-01

Vol. 2019 , num. 31-32, p. 5183-5186.

DOI : 10.1002/ejoc.201900500

“Doubly Orthogonal” Labeling of Peptides and Proteins

R. Tessier; J. Ceballos; N. Guidotti; R. Simonet-Davin; B. Fierz et al. 

Chem

2019-08-08

Vol. 5 , num. 8, p. 2243-2263.

DOI : 10.1016/j.chempr.2019.06.002

Ethynylbenziodazolones (EBZ) as Electrophilic Alkynylation Reagents for the Highly Enantioselective Copper-Catalyzed Oxyalkynylation of Diazo Compounds

D. P. Hari; L. Schouwey; V. Barber; R. Scopelliti; F. Fadaei-Tirani et al. 

Chemistry-A European Journal

2019-07-17

Vol. 25 , num. 40, p. 9522-9528.

DOI : 10.1002/chem.201900950

C-Terminal Bioconjugation of Peptides through Photoredox Catalyzed Decarboxylative Alkynylation

M. Garreau; F. Le Vaillant; J. Waser 

Angewandte Chemie-International Edition

2019-06-11

Vol. 58 , num. 24, p. 8182-8186.

DOI : 10.1002/anie.201901922

Stereoselective synthesis of alkyl-, aryl-, vinyl- and alkynyl-substituted Z-enamides and enol ethers

P. Caramenti; N. Declas; R. Tessier; M. D. Wodrich; J. Waser 

Chemical Science

2019-03-21

Vol. 10 , num. 11, p. 3223-3230.

DOI : 10.1039/c8sc05573d

Metal-Free Electrophilic Alkynylation of Sulfenate Anions with Ethynylbenziodoxolone Reagents

S. G. E. Amos; S. Nicolai; A. Gagnebin; F. Le Vaillant; J. Waser 

Journal Of Organic Chemistry

2019-03-15

Vol. 84 , num. 6, p. 3687-3701.

DOI : 10.1021/acs.joc.9b00050

Palladium-Catalyzed Carbo-Oxygenation of Propargylic Amines using in Situ Tether Formation

P. D. G. Greenwood; E. Grenet; J. Waser 

Chemistry-A European Journal

2019-02-26

Vol. 25 , num. 12, p. 3010-3013.

DOI : 10.1002/chem.201900020

Revisiting the Urech Synthesis of Hydantoins: Direct Access to Enantiopure 1,5-Substituted Hydantoins Using Cyanobenziodoxolone

N. Declas; F. Le Vaillant; J. Waser 

Organic Letters

2019-01-18

Vol. 21 , num. 2, p. 524-528.

DOI : 10.1021/acs.orglett.8b03843

2018

Cyclic Hypervalent Iodine Reagents for Azidation: Safer Reagents and Photoredox-Catalyzed Ring Expansion

S. Alazet; J. Preindl; R. Simonet-Davin; S. Nicolai; A. Nanchen et al. 

The Journal of Organic Chemistry

2018-09-15

Vol. 83 , num. 19, p. 12334-12356.

DOI : 10.1021/acs.joc.8b02068

Fine-Tuned Organic Photoredox Catalysts for Fragmentation-Alkynylation Cascades of Cyclic Oxime Ethers

F. Le Vaillant; M. Garreau; S. Nicolai; G. Gryn’ova; C. Corminboeuf et al. 

Chemical Science

2018-05-30

Vol. 9 , p. 5883-5889.

DOI : 10.1039/C8SC01818A

Rhodium-catalyzed C–H functionalization of heteroarenes using indoleBX hypervalent iodine reagents

E. Grenet; A. K. Das; P. Caramenti; J. Waser 

Beilstein Journal of Organic Chemistry

2018-05-25

Vol. 14 , p. 1208-1214.

DOI : 10.3762/bjoc.14.102

Metal-Free Oxidative Cross Coupling of Indoles with Electron-Rich (Hetero)arenes

P. Caramenti; R. Nandi; J. Waser 

Chemistry-A European Journal

2018-05-03

Vol. 24 , num. 40, p. 10049-10053.

DOI : 10.1002/chem.201802142

Iridium- and Rhodium-Catalyzed Directed C–H Heteroarylation of Benzaldehydes with Benziodoxolone Hypervalent Iodine Reagents

E. Grenet; J. Waser 

Organic Letters

2018-02-21

Vol. 20 , p. 1473-1476.

DOI : 10.1021/acs.orglett.8b00337

Lewis Acid Catalyzed Enantioselective Desymmetrization of Donor-Acceptor Meso-Diaminocyclopropanes

D. Perrotta; M. Wang; J. Waser 

Angewandte Chemie, International Edition

2018-02-20

Vol. 57 , p. 5120-5123.

DOI : 10.1002/anie.201800494

2017

Bench-Stable Electrophilic Indole and Pyrrole Reagents: Serendipitous Discovery and Use in C–H Functionalization

P. Caramenti 

Helvetica Chimica Acta

2017-10-30

Vol. 100 , p. e1700221.

DOI : 10.1002/hlca.201700221

Dearomatization of electron poor six-membered N-heterocycles through [3+2] annulation with aminocyclopropanes

J. Preindl; S. Chakrabarty; J. Waser 

Chemical Science

2017

Vol. 8 , num. 10, p. 7112-7118.

DOI : 10.1039/c7sc03197a

Indole- and Pyrrole-BX: Bench-Stable Hypervalent Iodine Reagents for Heterocycle Umpolung

P. Caramenti; S. Nicolai; J. Waser 

Chemistry-A European Journal

2017

Vol. 23 , num. 59, p. 14702-14706.

DOI : 10.1002/chem.201703723

Gold-catalyzed domino cyclization-alkynylation reactions with EBX reagents: new insights into the reaction mechanism

H. Ghari; Y. Li; R. Roohzadeh; P. Caramenti; J. Waser et al. 

Dalton Transactions

2017

Vol. 46 , num. 36, p. 12257-12262.

DOI : 10.1039/c7dt03154h

Enantioselective Copper-Catalyzed Oxy-Alkynylation of Diazo Compounds

D. P. Hari; J. Waser 

Journal Of The American Chemical Society

2017

Vol. 139 , num. 25, p. 8420-8423.

DOI : 10.1021/jacs.7b04756

Palladium-Catalyzed Carboamination of Allylic Alcohols Using a Trifluoroacetaldehyde-Derived Tether

B. Muriel; U. Orcel; J. Waser 

Organic Letters

2017

Vol. 19 , num. 13, p. 3548-3551.

DOI : 10.1021/acs.orglett.7b01524

Divergent Access to (1,1) and (1,2)-Azidolactones from Alkenes using Hypervalent Iodine Reagents

S. Alazet; F. Le Vaillant; S. Nicolai; T. Courant; J. Waser 

Chemistry-A European Journal

2017

Vol. 23 , num. 40, p. 9501-9504.

DOI : 10.1002/chem.201702599

Decarboxylative Alkynylation and Cyanation of Carboxylic Acids using Photoredox Catalysis and Hypervalent Iodine Reagents

F. Le Vaillant; J. Waser 

Chimia

2017

Vol. 71 , num. 4, p. 226-230.

DOI : 10.2533/chimia.2017.226

Room temperature decarboxylative cyanation of carboxylic acids using photoredox catalysis and cyanobenziodoxolones: a divergent mechanism compared to alkynylation

F. Le Vaillant; M. D. Wodrich; J. Waser 

Chemical Science

2017

Vol. 8 , num. 3, p. 1790-1800.

DOI : 10.1039/c6sc04907a

Heterotetracenes: Flexible Synthesis and in Silico Assessment of the Hole Transport Properties

Y. Li; G. Gryn’ova; F. Saenz; X. Jeanbourquin; K. Sivula et al. 

Chemistry A European Journal

2017

Vol. 23 , num. 33, p. 8058-8065.

DOI : 10.1002/chem.201701139

2016

One-Pot Three-Component Synthesis of Vicinal Diamines via In Situ Aminal Formation and Carboamination

U. Orcel; J. Waser 

Angewandte Chemie-International Edition

2016

Vol. 55 , num. 41, p. 12881-12885.

DOI : 10.1002/anie.201607318

Divergent Reactivity of Thioalkynes in Lewis Acid Catalyzed Annulations with Donor-Acceptor Cyclopropanes

S. Racine; B. Hegedus; R. Scopelliti; J. Waser 

Chemistry-A European Journal

2016

Vol. 22 , num. 34, p. 11997-12001.

DOI : 10.1002/chem.201602755

Nucleoside Analogues: Synthesis from Strained Rings

S. Racine; J. Vuilleumier; J. Waser 

Israel Journal Of Chemistry

2016

Vol. 56 , num. 6-7, p. 566-577.

DOI : 10.1002/ijch.201500090

Ethynyl benziodoxolones: functional terminators for cell-penetrating poly(disulfide)s

P. Morelli; X. Martin-Benlloch; R. Tessier; J. Waser; N. Sakai et al. 

Polymer Chemistry

2016

Vol. 7 , num. 20, p. 3465-3470.

DOI : 10.1039/c6py00562d

Gold-catalyzed direct alkynylation of tryptophan in peptides using TIPS-EBX

G. L. Tolnai; J. P. Brand; J. Waser 

Beilstein Journal Of Organic Chemistry

2016

Vol. 12 , p. 745-749.

DOI : 10.3762/bjoc.12.74

Copper-Catalyzed Oxy-Alkynylation of Diazo Compounds with Hypervalent Iodine Reagents

D. P. Hari; J. Waser 

Journal Of The American Chemical Society

2016

Vol. 138 , num. 7, p. 2190-2193.

DOI : 10.1021/jacs.6b00278

Alkynylation of Thiols with Ethynylbenziodoxolone (EBX) Reagents: alpha- or beta- pi-Addition?

M. D. Wodrich; P. Caramenti; J. Waser 

Organic Letters

2016

Vol. 18 , num. 1, p. 60-63.

DOI : 10.1021/acs.orglett.5b03241

2015

Enantioselective Synthesis of Homoallylic Azides and Nitriles via Palladium-Catalyzed Decarboxylative Allylation

M. V. Vita; P. Caramenti; J. Waser 

Organic Letters

2015

Vol. 17 , num. 23, p. 5832-5835.

DOI : 10.1021/acs.orglett.5b03002

Room-Temperature Decarboxylative Alkynylation of Carboxylic Acids Using Photoredox Catalysis and EBX Reagents

F. Le Vaillant; T. Courant; J. Waser 

Angewandte Chemie-International Edition

2015

Vol. 54 , num. 38, p. 11200-11204.

DOI : 10.1002/anie.201505111

Platinum-Catalyzed Domino Reactionwith Benziodoxole Reagents for Accessing Benzene-Alkynylated Indoles

Y. Li; J. Waser 

Angewandte Chemie-International Edition

2015

Vol. 54 , num. 18, p. 5438-5442.

DOI : 10.1002/anie.201412321

Cyclic Hypervalent Iodine Reagents and Iron Catalysts: The Winning Team for Late-Stage C-H Azidation

M. V. Vita; J. Waser 

Angewandte Chemie-International Edition

2015

Vol. 54 , num. 18, p. 5290-5292.

DOI : 10.1002/anie.201501666

In the Lab Combining Catalyst and Reagent Design for Electrophilic Alkynylation Johnson Matthey Technology Review features new laboratory research

J. Waser 

Johnson Matthey Technology Review

2015

Vol. 59 , num. 3, p. 284-286.

DOI : 10.1595/205651315X688587

Intramolecular palladium-catalyzed alkene carboalkynylation

S. Nicolai; P. Swallow; J. Waser 

Tetrahedron

2015

Vol. 71 , num. 35, p. 5959-5964.

DOI : 10.1016/j.tet.2015.06.030

Proteome-Wide Profiling of Targets of Cysteine reactive Small Molecules by Using Ethynyl Benziodoxolone Reagents

D. Abegg; R. Frei; L. Cerato; D. P. Hari; C. Wang et al. 

Angewandte Chemie-International Edition

2015

Vol. 54 , num. 37, p. 10852-10857.

DOI : 10.1002/anie.201505641

1-Alkynyltriazenes as Functional Analogues of Ynamides

F. G. Perrin; G. Kiefer; L. Jeanbourquin; S. Racine; D. Perrotta et al. 

Angewandte Chemie -International Edition in English-

2015

Vol. 54 , p. 13393-13396.

DOI : 10.1002/anie.201507033

General and Practical Formation of Thiocyanates from Thiols

R. Frei; T. Courant; M. D. Wodrich; J. Waser 

Chemistry-A European Journal

2015

Vol. 21 , num. 6, p. 2662-2668.

DOI : 10.1002/chem.201406171

One-Pot, Three-Component Arylalkynyl Sulfone Synthesis

C. C. Chen; J. Waser 

Organic Letters

2015

Vol. 17 , num. 3, p. 736-739.

DOI : 10.1021/acs.orglett.5b00015

Palladium-Catalyzed Vicinal Amino Alcohols Synthesis from Allyl Amines by In Situ Tether Formation and Carboetherification

U. Orcel; J. Waser 

Angewandte Chemie-International Edition

2015

Vol. 54 , num. 17, p. 5250-5254.

DOI : 10.1002/anie.201500636

[4+2]-Annulations of Aminocyclobutanes

D. Perrotta; S. Racine; J. Vuilleumier; F. De Nanteuil; J. Waser 

Organic Letters

2015

Vol. 17 , num. 4, p. 1030-1033.

DOI : 10.1021/acs.orglett.5b00149

2014

Fast and Highly Chemoselective Alkynylation of Thiols with Hypervalent Iodine Reagents Enabled through a Low Energy Barrier Concerted Mechanism

R. Frei; M. D. Wodrich; D. P. Hari; P-A. Bonin; C. Chauvier et al. 

Journal Of The American Chemical Society

2014

Vol. 136 , num. 47, p. 16563-16573.

DOI : 10.1021/ja5083014

Enantioselective Synthesis of Polycyclic Carbocycles via an Alkynylation-Allylation-Cyclization Strategy

M. V. Vita; P. Mieville; J. Waser 

Organic Letters

2014

Vol. 16 , num. 21, p. 5768-5771.

DOI : 10.1021/ol5028333

Diester-Substituted Aminocyclopropanes: Synthesis and Use in [3+2]-Annulation Reactions

E. Serrano; F. De Nanteuil; J. Waser 

Synlett

2014

Vol. 25 , num. 16, p. 2285-2288.

DOI : 10.1055/s-0034-1378512

Room temperature alkynylation of H-phosphi(na)tes and secondary phosphine oxides with ethynylbenziodoxolone (EBX) reagents

C. C. Chen; J. Waser 

Chemical Communications

2014

Vol. 50 , num. 85, p. 12923-12926.

DOI : 10.1039/c4cc06851c

Cyclization and annulation reactions of nitrogen-substituted cyclopropanes and cyclobutanes

F. De Nanteuil; F. De Simone; R. Frei; F. Benfatti; E. Serrano et al. 

Chemical Communications

2014

Vol. 50 , num. 75, p. 10912-10928.

DOI : 10.1039/c4cc03194f

Synthesis of (Carbo) nucleoside Analogues by [3+2] Annulation of Aminocyclopropanes

S. Racine; F. De Nanteuil; E. Serrano; J. Waser 

Angewandte Chemie-International Edition

2014

Vol. 53 , num. 32, p. 8484-8487.

DOI : 10.1002/anie.201404832

Dynamic Kinetic Asymmetric [3+2] Annulation Reactions of Aminocyclopropanes

F. De Nanteuil; E. Serrano; D. Perrotta; J. Waser 

Journal Of The American Chemical Society

2014

Vol. 136 , num. 17, p. 6239-6242.

DOI : 10.1021/ja5024578

2013

Total Synthesis and Biological Evaluation of Jerantinine E

R. Frei; D. Städler; A. Raja; R. Franke; F. Sasse et al. 

Angewandte Chemie -International Edition in English-

2013

Vol. 52 , num. 50, p. 13373-13376.

DOI : 10.1002/anie.201305533

Gold-Catalyzed Regioselective Synthesis of 2- and 3-Alkynyl Furans

Y. Li; J. P. Brand; J. Waser 

Angewandte Chemie-International Edition

2013

Vol. 52 , num. 26, p. 6743-6747.

DOI : 10.1002/anie.201302210

A Highly Chemoselective and Practical Alkynylation of Thiols

R. Frei; J. Waser 

Journal Of The American Chemical Society

2013

Vol. 135 , num. 26, p. 9620-9623.

DOI : 10.1021/ja4044196

Azidation of beta-Keto Esters and Silyl Enol Ethers with a Benziodoxole Reagent

M. V. Vita; J. Waser 

Organic Letters

2013

Vol. 15 , num. 13, p. 3246-3249.

DOI : 10.1021/ol401229v

Catalytic Friedel-Crafts Reaction of Aminocyclopropanes

F. De Nanteuil; J. Loup; J. Waser 

Organic Letters

2013

Vol. 15 , num. 14, p. 3738-3741.

DOI : 10.1021/ol401616a

Synthesis of Aminocyclobutanes by Iron-Catalyzed [2+2] Cycloaddition

F. De Nanteuil; J. Waser 

Angewandte Chemie-International Edition

2013

Vol. 52 , num. 34, p. 9009-9013.

DOI : 10.1002/anie.201303803

Zinc-gold cooperative catalysis for the direct alkynylation of benzofurans

Y. Li; J. Waser 

Beilstein Journal Of Organic Chemistry

2013

Vol. 9 , p. 1763-1767.

DOI : 10.3762/bjoc.9.204

Pd(0)-Catalyzed Alkene Oxy- and Aminoalkynylation with Aliphatic Bromoacetylenes

S. Nicolai; R. Sedigh-Zadeh; J. Waser 

Journal Of Organic Chemistry

2013

Vol. 78 , num. 8, p. 3783-3801.

DOI : 10.1021/jo400254q

Ethynylbenziodoxolones (EBX) as Reagents for the Ethynylation of Stabilized Enolates

D. F. Gonzalez; J. P. Brand; R. Mondiere; J. Waser 

Advanced Synthesis & Catalysis

2013

Vol. 355 , num. 8, p. 1631-1639.

DOI : 10.1002/adsc.201300266

C2-Selective Direct Alkynylation of Indoles

G. L. Tolnai; S. Ganss; J. P. Brand; J. Waser 

Organic Letters

2013

Vol. 15 , num. 1, p. 112-115.

DOI : 10.1021/ol3031389

2012

Ethynyl Benziodoxolones for the Direct Alkynylation of Heterocycles: Structural Requirement, Improved Procedure for Pyrroles, and Insights into the Mechanism

J. P. Brand; C. Chevalley; R. Scopelliti; J. Waser 

Chemistry-A European Journal

2012

Vol. 18 , p. 5655-5666.

DOI : 10.1002/chem.201200200

Synthesis of 1-[(Triisopropylsilyl)ethynyl]-1 lambda(3),2-benziodoxol-3(1H)-one and Alkynylation of Indoles, Thiophenes, and Anilines

J. P. Brand; J. Waser 

Synthesis-Stuttgart

2012

Vol. 44 , p. 1155-1158.

DOI : 10.1055/s-0031-1290589

Catalytic Enantiospecific [3+2] Annulation of Aminocyclopropanes with Ketones

F. Benfatti; F. de Nanteuil; J. Waser 

Chemistry-A European Journal

2012

Vol. 18 , p. 4844-4849.

DOI : 10.1002/chem.201103971

Para-Selective Gold-Catalyzed Direct Alkynylation of Anilines

J. P. Brand; J. Waser 

Organic Letters

2012

Vol. 14 , p. 744-747.

DOI : 10.1021/ol203289v

Iron-Catalyzed [3+2] Annulation of Aminocyclopropanes with Aldehydes: Stereoselective Synthesis of Aminotetrahydrofurans

F. Benfatti; F. de Nanteuil; J. Waser 

Organic Letters

2012

Vol. 14 , p. 386-389.

DOI : 10.1021/ol203144v

2011

Formal Homo-Nazarov and Other Cyclization Reactions of Activated Cyclopropanes

F. De Simone; T. Saget; F. Benfatti; S. Almeida; J. Waser 

Chemistry – A European Journal

2011

Vol. 17 , num. 51, p. 14527-14538.

DOI : 10.1002/chem.201102583

Catalytic [3+2] Annulation of Aminocyclopropanes for the Enantiospecific Synthesis of Cyclopentylamines

F. de Nanteuil; J. Waser 

Angewandte Chemie, International Edition

2011

Vol. 50 , num. 50, p. 12075-12079.

DOI : 10.1002/anie.201106255

Benziodoxole-based hypervalent iodine reagents for atom-transfer reactions

J. P. Brand; D. Gonzalez Fernandez; S. Nicolai; J. Waser 

Chemical Communications

2011

Vol. 47 , p. 102-115.

DOI : 10.1039/c0cc02265a

One-pot gold-catalyzed synthesis of 3-silylethynyl indoles from unprotected o-alkynylanilines

J. P. Brand; C. Chevalley; J. Waser 

Beilstein Journal Of Organic Chemistry

2011

Vol. 7 , p. 565-569.

DOI : 10.3762/bjoc.7.65

Cyclopropanes and Hypervalent Iodine Reagents: High Energy Compounds for Applications in Synthesis and Catalysis

D. Gonzalez Fernandez; F. De Simone; J. P. Brand; S. Nicolai; J. Waser 

Chimia

2011

Vol. 65 , p. 649-651.

DOI : 10.2533/chimia.2011.649

Pd(0)-Catalyzed Oxy- and Aminoalkynylation of Olefins for the Synthesis of Tetrahydrofurans and Pyrrolidines

S. Nicolai; J. Waser 

Organic Letters

2011

Vol. 13 , p. 6324-6327.

DOI : 10.1021/ol2029383

A Palladium-Catalyzed Aminoalkynylation Strategy towards Bicyclic Heterocycles: Synthesis of (±)-Trachelanthamidine

S. Nicolai; C. Piemontesi; J. Waser 

Angewandte Chemie, International Edition

2011

Vol. 50 , num. 20, p. 4680-4683.

DOI : 10.1002/anie.201100718

2010

Direct Alkynylation of Thiophenes: Cooperative Activation of TIPS–EBX with Gold and Brønsted Acids

J. P. Brand; J. Waser 

Angewandte Chemie, International Edition

2010

Vol. 49 , num. 40, p. 7304-7307.

DOI : 10.1002/anie.201003179

Ethynyl-1,2-benziodoxol-3(1 H)-one (EBX): An Exceptional Reagent for the Ethynylation of Keto, Cyano, and Nitro Esters

D. Fernández González; J. P. Brand; J. Waser 

Chemistry, A European Journal

2010

Vol. 16 , num. 31, p. 9457-9461.

DOI : 10.1002/chem.201001539

Catalytic Selective Cyclizations of Aminocyclopropanes: Formal Synthesis of Aspidospermidine and Total Synthesis of Goniomitine

F. De Simone; J. Gertsch; J. Waser 

Angewandte Chemie, International Edition

2010

Vol. 49 , p. 5767-5770.

DOI : 10.1002/anie.201001853

Synthesis of Chiral Bifunctional (Thio)Urea N-Heterocyclic Carbenes

J. P. Brand; J. I. Osuna-Siles; J. Waser 

Synlett

2010

p. 881-884.

DOI : 10.1055/s-0029-1219543

Pd-Catalyzed Intramolecular Oxyalkynylation of Alkenes with Hypervalent Iodine

S. Nicolai; S. Erard; D. Fernandez Gonzalez; J. Waser 

Organic Letters

2010

Vol. 12 , num. 2, p. 384-387.

DOI : 10.1021/ol9027286

2009

Direct Alkynylation of Indole and Pyrrole Heterocycles

J. P. Brand; J. Charpentier; J. Waser 

Angewandte Chemie, International Edition

2009

Vol. 48 , num. 49, p. 9346-9349.

DOI : 10.1002/anie.200905419

Catalytic Formal Homo-Nazarov Cyclization

F. De Simone; J. Andrès; R. Torosantucci; J. Waser 

Organic Letters

2009

Vol. 11 , num. 4, p. 1023-1026.

DOI : 10.1021/ol802970g

2008

Total Synthesis of (-)-Pseudolaric Acid B

B. M. Trost; J. Waser; A. Meyer 

Journal of the American Chemical Society

2008

Vol. 130 , num. 48, p. 16424-16434.

DOI : 10.1021/ja806724x

2007

Cobalt-Catalyzed Synthesis of Tertiary Azides from α,α-Disubstituted Olefins under Mild Conditions Using Commercially Available Reagents

B. Gaspar; J. Waser; E. M. Carreira 

Synthesis

2007

num. 24, p. 3839-3845.

Total synthesis of (-)-pseudolaric Acid B

B. M. Trost; J. Waser; A. Meyer 

Journal of the American Chemical Society

2007

Vol. 129 , num. 47, p. 14556-7.

DOI : 10.1021/ja076165q

2006

Hydrazines and Azides via the Metal-Catalyzed Hydrohydrazination and Hydroazidation of Olefins

J. Waser; B. Gaspar; H. Nambu; E. M. Carreira 

Journal of the American Chemical Society

2006

Vol. 128 , num. 35, p. 11693-11712.

DOI : 10.1021/ja062355+

2005

Cobalt-Catalyzed Hydrohydrazination of Dienes and Enynes: Access to Allylic and Propargylic Hydrazides

J. Waser; J. C. Gonzalez-Gomez; H. Nambu; P. Huber; E. M. Carreira 

Organic Letters

2005

Vol. 7 , num. 19, p. 4249-4252.

DOI : 10.1021/ol0517473

Cobalt-Catalyzed Hydroazidation of Olefins: Convenient Access to Alkyl Azides

J. Waser; H. Nambu; E. M. Carreira 

Journal of the American Chemical Society

2005

Vol. 127 , num. 23, p. 8294-8295.

DOI : 10.1021/ja052164r

2004

Alkene hydrazination: Catalytic hydrohydrazination of a wide range of alkenes with a simple Mn complex

J. Waser; E. M. Carreira 

Angewandte Chemie, International Edition

2004

Vol. 43 , num. 31, p. 4099-4102.

DOI : 10.1002/anie.200460811

Convenient synthesis of alkylhydrazides by the cobalt-catalyzed hydrohydrazination reaction of olefins and azodicarboxylates

J. Waser; E. M. Carreira 

Journal of the American Chemical Society

2004

Vol. 126 , num. 18, p. 5676-5677.

DOI : 10.1021/ja048698u

2001

Synthetic process development and scale up of palladium-catalyzed alkoxycarbonylation of chloropyridines

R. Crettaz; J. Waser; Y. Bessard 

Organic Process Research & Development

2001

Vol. 5 , num. 6, p. 572-574.

DOI : 10.1021/op010012k

Reviews

2018

Cyclic Hypervalent Iodine Reagents: Enabling Tools for Bond Disconnection via Reactivity Umpolung

D. P. Hari; P. Caramenti; J. Waser 

Accounts of Chemical Research

2018-11-28

Vol. 51 , num. 12, p. 3212-3225.

DOI : 10.1021/acs.accounts.8b00468

2017

In situ tether formation from amines and alcohols enabling highly selective Tsuji-Trost allylation and olefin functionalization

U. Orcel; J. Waser 

Chemical Science

2017

Vol. 8 , num. 1, p. 32-39.

DOI : 10.1039/c6sc04366f

2016

Benziodoxol(on)e Reagents as Tools in Organic Synthesis: The Background behind the Discovery at the Laboratory of Catalysis and Organic Synthesis

J. Waser 

Synlett

2016

Vol. 27 , num. 20, p. 2761-2773.

DOI : 10.1055/s-0036-1589409

Cyclic Hypervalent Iodine Reagents for Atom-Transfer Reactions: Beyond Trifluoromethylation

Y. Li; D. P. Hari; M. V. Vita; J. Waser 

Angewandte Chemie-International Edition

2016

Vol. 55 , num. 14, p. 4436-4454.

DOI : 10.1002/anie.201509073

2014

Taming Hypervalent Bonds and Strained Rings for Catalysis and Synthesis

F. De Nanteuil; Y. Li; M. V. Vita; R. Frei; E. Serrano et al. 

Chimia

2014

Vol. 68 , num. 7-8, p. 516-521.

DOI : 10.2533/chimia.2014.516

2013

Gold-Catalyzed Alkynylation: Acetylene-Transfer instead of Functionalization

J. P. Brand; Y. Li; J. Waser 

Israel Journal Of Chemistry

2013

Vol. 53 , num. 11-12, p. 901-910.

DOI : 10.1002/ijch.201300044

2012

Asymmetric Organocatalysis Meets Hypervalent Iodine Chemistry for the alpha-Functionalization of Carbonyl Compounds

D. Gonzalez Fernandez; F. Benfatti; J. Waser 

Chemcatchem

2012

Vol. 4 , p. 955-958.

DOI : 10.1002/cctc.201200116

Indole Alkaloids Synthesis via a Selective Cyclization of Aminocyclopropanes

F. De Simone; J. Waser 

Chimia

2012

Vol. 66 , p. 233-236.

DOI : 10.2533/chimia.2012.233

Electrophilic alkynylation: the dark side of acetylene chemistry

J. P. Brand; J. Waser 

Chemical Society Reviews

2012

Vol. 41 , p. 4165-4179.

DOI : 10.1039/c2cs35034c

2011

Cyclization of Aminocyclopropanes in Indole Alkaloids Synthesis

F. De Simone; J. Waser 

Synlett

2011

num. 5, p. 589-593.

DOI : 10.1055/s-0030-1259553

Benziodoxole-based hypervalent iodine reagents for atom-transfer reactions

J. P. Brand; D. Fernandez Gonzalez; S. Nicolai; J. Waser 

Chemical Communications- Royal Society of Chemistry

2011

Vol. 47 , p. 102-115.

DOI : 10.1039/C0CC02265A

2009

Cyclization and Cycloaddition Reactions of Cyclopropyl Carbonyls and Imines

F. De Simone; J. Waser 

Synthesis

2009

num. 20, p. 3353-3374.

DOI : 10.1055/s-0029-1216998

Cyclization of Cyclopropyl Carbonyls and the Homo-Nazarov Reaction

F. De Simone; J. Waser 

Chimia

2009

Vol. 63 , num. 3, p. 162-167.

DOI : 10.2533/chimia.2009.162

Theses

2019

Development of New Strategies of Umpolung with Cyclic Hypervalent Iodine Reagents

P. Caramenti / Director(s) : J. Waser 

Lausanne: EPFL

2019

p. 598.

DOI : 10.5075/epfl-thesis-9502

Photoredox-Catalyzed Decarboxylation for the Transfer of Alkynes and Nitriles Using Hypervalent Iodine Reagents

F. Le Vaillant / Director(s) : J. Waser 

Lausanne: EPFL

2019

p. 448.

DOI : 10.5075/epfl-thesis-9212

Application of Hypervalent Iodine Reagents for Novel Cysteine Labeling

R. G. Tessier / Director(s) : J. Waser 

Lausanne: EPFL

2019

p. 443.

DOI : 10.5075/epfl-thesis-9119

2018

Developing Reactions of Strained Rings

D. Perrotta / Director(s) : J. Waser 

Lausanne: EPFL

2018

p. 332.

DOI : 10.5075/epfl-thesis-8579

2017

In Situ Tethering Strategies for the 3-Component Synthesis of Vicinal Amino Alcohols and Diamines via Pd-Catalyzed Carboetherification and Carboamination

U. J. Orcel / Director(s) : J. Waser 

Lausanne: EPFL

2017

p. 328.

DOI : 10.5075/epfl-thesis-7319

2016

Lewis acid Catalyzed Annulations of Donor-Acceptor Aminocyclopropanes and Aminocyclobutanes

S. L. Racine / Director(s) : J. Waser 

Lausanne: EPFL

2016

p. 478.

DOI : 10.5075/epfl-thesis-7199

Synthesis of Alkynylated Heterocycles by Direct C-H Alkynylation or Domino Alkynylation Reactions

Y. Li / Director(s) : J. Waser 

Lausanne: EPFL

2016

p. 356.

DOI : 10.5075/epfl-thesis-6915

2015

Cyclic Hypervalent Iodine Reagents and Pd-Catalysis

M. V. Vita / Director(s) : J. Waser 

Lausanne: EPFL

2015

p. 846.

DOI : 10.5075/epfl-thesis-6624

2014

Synthesis and Reactivity of Donor-Acceptor Substituted Aminocyclopropanes and Aminocyclobutanes

F. de Nanteuil / Director(s) : J. Waser 

Lausanne: EPFL

2014

DOI : 10.5075/epfl-thesis-6268

2013

Pd-Catalyzed Oxy- and Aminoalkynylation of Olefins

S. Nicolai / Director(s) : J. Waser 

Lausanne: EPFL

2013

DOI : 10.5075/epfl-thesis-5620

2012

Development of Catalytic Umpolung

J. Brand / Director(s) : J. Waser 

Lausanne: EPFL

2012

DOI : 10.5075/epfl-thesis-5397

Catalytic Formal Homo-Nazarov Reaction and Other Cyclizations of Cyclopropanes

F. De Simone / Director(s) : J. Waser 

Lausanne: EPFL

2012

p. 350.

DOI : 10.5075/epfl-thesis-5269

2011

New Acetylene Chemistry

D. Fernández González / Director(s) : J. Waser 

Lausanne: EPFL

2011

p. 294.

DOI : 10.5075/epfl-thesis-5214

Book Chapters

2018

Alkynylations and Vinylations

D. P. Hari; S. Nicolai; J. Waser 

PATAI’S Chemistry of Functional Groups; Wiley, 2018-06-13. p. 1-58.

DOI : 10.1002/9780470682531.pat0951

2015

Alkynylation with Hypervalent Iodine Reagents

J. Waser 

Hypervalent Iodine Chemistry; Springer Verlag, 2015. p. 187-222.

ISBN : 978-3-319-33733-3

DOI : 10.1007/128_2015_660

2013

Synthesis of Saturated Heterocycles via Metal-Catalyzed Formal Cycloaddition Reactions That Generate a C–N or C–O Bond

J. Waser 

Synthesis of Heterocycles via Metal-Catalyzed Reactions that Generate One or More Carbon-Heteroatom Bonds; Berlin Heidelberg: Springer Verlag, 2013. p. 225-270.

ISBN : 978-3-642-38879-8

DOI : 10.1007/7081_2013_108

2010

Azides by Olefin Hydroazidation Reactions

J. Waser; E. M. Carreira 

Organic Azides: Syntheses and Applications; Wiley, 2010. p. 95-112.