Publications

Journal Articles

2024

SOMOphilic alkyne vs radical-polar crossover approaches: The full story of the azido-alkynylation of alkenes
Julien Borrel and Jerome Waser
Beilstein J. Org. Chem. 2024, 20, 701-713. (10.3762/bjoc.20.64) Open Access!

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Benzylic C(sp3)−H Azidation: Copper vs Iron Catalysis
Angel Rentería-Gómez, Rubén O. Torres-Ochoa, Pierre Palamini, Raphaël Simonet-Davin, Qian Wang, Jérôme Waser, Jieping Zhu
Helv. Chim. Acta 2024, 107, e202400004. (10.1002/hlca.202400004) Open Access!

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Interrupted Polonovski Strategy for the Synthesis of Functionalized Amino Acids and Peptides
Christine Marty, Emmanuelle M. D. Allouche, and Jerome Waser
Org. Lett. 2024, 26, 456-460. (10.1021/acs.orglett.3c03603) Green Access Raw data

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2023

Synthesis of Fluorescent Cyclic Peptides via Gold(I)-Catalyzed Macrocyclization
Xing-Yu Liu, Wei Cai, Nathan Ronceray, Aleksandra Radenovic, Beat Fierz and Jerome Waser
J. Am. Chem. Soc. 2023, 145, 26525-26531. (10.1021/jacs.3c09261) Open Access! Raw data

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Photocatalyzed [2σ + 2σ] and [2σ + 2π] Cycloadditions for the Synthesis of Bicyclo[3.1.1]heptanes and 5- or 6-Membered Carbocycles
Tin V. T. Nguyen, André Bossonnet, Matthew D. Wodrich and Jerome Waser
J. Am. Chem. Soc. 2023, 145, 25411-25421. (10.1021/jacs.3c09789) Green Access Raw data

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Acyl-Ethynylbenziodoxolone (acyl-EBX): Access to Ketene Dithioarylacetals
Pierre Palamini, Julien Borrel, Maël Djaïd, Morgane Delattre and Jerome Waser
Org. Lett. 2023, 25, 7535-7539. (10.1021/acs.orglett.3c02869) Green Access Raw data

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One-pot synthesis of functionalized bis(trifluoromethylated)benziodoxoles from iodine(i) precursors
Tobias M. Milzarek, Nieves P. Ramirez, Xing-Yu Liu and Jerome Waser
Chem. Commun. 2023, 59, 12637-12640. (10.1039/D3CC04525K) Green Access Raw data

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Cysteine-Cysteine Cross-Conjugation of both Peptides and Proteins with a Bifunctional Hypervalent Iodine-Electrophilic Reagent
Ilias Koutsopetras, Abhaya Kumar Mishra, Rania Benazza, Oscar Hernandez-Alba, Sarah Cianférani, Guilhem Chaubet, Stefano Nicolai and Jerome Waser
Chem. Eur. J. 2023, 29, e202302689. (10.1002/chem.202302689) Open Access!

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Semipinacol Rearrangement of Cyclopropenylcarbinols for the Synthesis of Highly Substituted Cyclopropanes
Vladyslav Smyrnov and Jerome Waser
Org. Lett. 2023, 25, 6999-7003. (10.1021/acs.orglett.3c02543) Green Access Raw data

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Iron-Catalyzed Synthesis of α-Azido α-Amino Esters via the Alkylazidation of Alkenes
Pierre Palamini, Emmanuelle M. D. Allouche, and Jerome Waser
Org. Lett. 2023, 25, 6791-6795. (DOI: 10.1021/acs.orglett.3c02153) Open Access! Raw data

Azido-alkynylation of alkenes through radical-polar crossover
Julien Borrel and Jerome Waser
Chem. Sci. 2023, 14, 9452-9460. (DOI: 10.1039/D3SC03309K) Open Access! Raw data

Photochemical [2+2] Cycloaddition of Alkynyl Boronates
Oleksandr S. Liashuk, Oleksandr O. Grygorenko, Yulian M. Volovenko and Jerome Waser
Chem. Eur. J. 2023, 29, e202301650. (DOI: 10.1002/chem.202301650) Open Access! Raw data

Synthesis of Trifluoromethylated Alkenes: Hypervalent Iodine Meets High-Valent Copper
Tobias Michael Milzarek and Jerome Waser
Angew. Chem., Int. Ed. 2023, 62, e202306128. (DOI: 10.1002/anie.202306128) Open Access! Raw data

Peptide-Hypervalent Iodine Reagent Chimeras: Enabling Peptide Functionalization and Macrocyclization
Xing-Yu Liu, Xinjian Ji, Christian Heinis and Jerome Waser
Angew. Chem., Int. Ed. 2023, 62, e202306036. (DOI: 10.1002/anie.202306036) Open Access! Raw data

Copper (I)-BOX Catalyzed Asymmetric 3-Component Reaction for the Synthesis of Trifluoromethylated Propargylic Ethers and Anilines
Nieves P. Ramirez and Jerome Waser
Angew. Chem., Int. Ed. 2023, 62, e202305776. (DOI: 10.1002/anie.202305776) Open Access! Raw data

Synthesis of propargyl silanes from terminal alkynes via a migratory Sonogashira reaction
Mikus Purins, Lucas Eichenberger, and Jerome Waser
Chem. Commun. 2023, 59, 7931-7934. (DOI: 10.1039/D3CC01847D ) Open Access! Raw data

Donor-Acceptor Aminocyclobutane Monoesters: Synthesis and Silylium-Catalyzed (4+2) Annulation with Indoles
Emma G. L. Robert, Vincent Pirenne, Matthew D. Wodrich and Jerome Waser
Angew. Chem., Int. Ed. 2023, 62, e202302420. (DOI: 10.1002/anie.202302420 ) Open Access! Raw data

X-Ray and NMR Structural Data of Ethynylbenziodoxolones (EBXs) Reagents and Their Analogues
Eliott Le Du, Nieves P. Ramirez, Stefano Nicolai, Rosario Scopelliti, Farzaneh Fadaei-Tirani, Matthew D. Wodrich, Durga Prasad Hari and Jerome Waser
Helv. Chim. Acta 2023, e202200175. (DOI: 10.1002/hlca.202200175 ) Open Access!

Review Articles

2023

Recent progress in alkynylation with hypervalent iodine reagents
Eliott Le Du and Jerome Waser
Chem. Commun. 2023, 59, 1589-1604. (DOI: 10.1039/D2CC06168F ) Open Access!

Publications prior to 2023

Publications 2020-2022
Publications 2017-2019
Publications 2013-2016
Publications 2009-2012