Publications

Journal Articles

2021

Cys‐Cys and Cys‐Lys Stapling of Unprotected Peptides Enabled by Hypervalent Iodine Reagents
Javier Ceballos, Elija Grinhagena, Gontran Sangouard, Christian Heinis and Jerome Waser
Angew. Chem., Int. Ed. 2021, in press. (10.1002/anie.202014511)

Collaboration: The binding affinity of the stapled peptides was measured at the Heinis group .

Small peptide diversification through photoredox-catalyzed oxidative C-terminal modification
Eliott Le Du, Marion Garreau and Jerome Waser
Chem. Sci. 2021, 12, 2467-2473. (10.1039/d0sc06180h) Raw data

2020

Low‐Temperature Intramolecular [4+2] Cycloaddition of Allenes with Arenes for the Synthesis of Diene Ligands
Durga Prasad Hari, Guillaume Pisella, Matthew D. Wodrich, Artem V. Tsymbal, Farzaneh Fadaei Tirani, Rosario Scopelliti and Jerome Waser
Angew. Chem., Int. Ed. 2021, 60, 5475-5481. (10.1002/anie.202012299)

Azide Radical Initiated Ring Opening of Cyclopropenes Leading to Alkenyl Nitriles and Polycyclic Aromatic Compounds
Bastian Muriel and Jerome Waser
Angew. Chem., Int. Ed. 2021, 60, 4075-4079. (10.1002/anie.202013516) Raw data

Synthesis of Thiochromans via [3+3] Annulation of Aminocyclopropanes with Thiophenols
Ming-Ming Wang, Seongmin Jeon and Jerome Waser
Org. Lett. 2020, 22, 9123-9127. (10.1021/acs.orglett.0c03528) Raw data

Enantioselective Carboetherification/Hydrogenation for the Synthesis of Amino Alcohols via a Catalytically Formed Chiral Auxiliary
Luca Buzzetti, Mikus Purins, Phillip D. G. Greenwood and Jerome Waser
J. Am. Chem. Soc. 2020, 142, 17334-17339. (10.1021/jacs.0c09177 ) Raw data

Photocatalytic Umpolung of N- and O- Substituted Alkenes for the Synthesis of 1,2-Amino Alcohols and Diols
Stephanie G. E. Amos, Stefano Nicolai and Jerome Waser
Chem. Sci. 2020, 11, 11274-11279. (10.1039/D0SC03655B ) Raw data

Photochemical Functionalization of Heterocycles with EBX Reagents; C‐H Alkynylation versus Deconstructive Ring Cleavage
Errika Voutyritsa, Marion Garreau, Maroula G. Kokotou, Ierasia Triandafillidi, Jérôme Waser and Christoforos G. Kokotos
Chem. Eur. J. 2020, 26, 14453-14460. (10.1002/chem.202002868 )

Collaboration: The photoredox chemistry was developed at the Kokotos group .

Oxidative Fluorination of Cyclopropylamides via Organic Photoredox Catalysis
Ming-Ming Wang and Jerome Waser
Angew. Chem., Int. Ed. 2020, 59, 16420-16424. (10.1002/anie.202007864 ) Raw data Green Access

Access to Vinyl Ethers and Ketones with Hypervalent Iodine Reagents as Oxy‐Allyl Cation Synthetic Equivalents
Nina Declas and Jerome Waser
Angew. Chem., Int. Ed. 2020, 59, 18256-18260. (10.1002/anie.202006707 ) Raw data Green Access

Triazene-Activated Donor–Acceptor Cyclopropanes: Ring-Opening and (3 + 2) Annulation Reactions
Abdusalom A. Suleymanov, Eliott Le Du, Zhaowen Dong, Bastian Muriel, Rosario Scopelliti, Farzaneh Fadaei-Tirani, Jérôme Waser and Kay Severin
Org. Lett. 2020, 22, 10, 4517-4522. (10.1021/acs.orglett.0c01527 ) Raw data Green Access

Collaboration: The triazene chemistry was developed at the Severin group .

Copper-Catalyzed Oxyvinylation of Diazo Compounds
Guillaume Pisella, Alec Gagnebin and Jerome Waser
Org. Lett. 2020, 22, 10, 3884–3889. (10.1021/acs.orglett.0c01150 ) Raw data Green Access

Ethynylation of Cysteines from Peptides to Proteins in Living Cells
Romain Tessier, Raj Kumar Nandi, Brendan G. Dwyer, Daniel Abegg, Charlotte Sornay, Javier Ceballos, Stephane Erb, Sarah Cianferani, Alain Wagner, Guilhem Chaubet and Jerome Waser
Angew. Chem., Int. Ed. 2020, 59, 10961-10970. (10.1002/anie.202002626 ) Green Access

Collaboration: Antibody modification studies were done in the Wagner/Chaubet group and proteomic studies were done in the Adibekian group .

Three‐Component Reaction for the Synthesis of Highly Functionalized Propargyl Ethers
Guillaume Pisella, Alec Gagnebin and Jerome Waser
Chem. Eur. J. 2020, 26, 10199-10204. (DOI:10.1002/chem.202001317 ) Green Access

Copper-Catalyzed Oxyalkynylation of C–S Bonds in Thiiranes and Thiethanes with Hypervalent Iodine Reagents
Julien Borrel, Guillaume Pisella and Jerome Waser
Org. Lett. 2020, 22, 422-427. (DOI:10.1021/acs.orglett.9b04157 ) Raw data Green Access

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One-Pot Synthesis of 1-[(Triisopropylsilyl)ethynyl]-1,2-benziodoxol-3(1H)-one (TIPS-EBX): Process Safety Assessment and Impact of Impurities on Product Stability
Durga Prasad Hari, Paola Caramenti, Lionel Schouwey, Miyeon Chang, Stefano Nicolai, Donald Bachert, Timothy Wright, Chuck Orella and Jerome Waser
Org. Process Res. Dev. 2020, 24, 106-110. (DOI:10.1021/acs.oprd.9b00498 ) Green Access

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Review Articles

2020

Palladium-Catalyzed Functionalization of Olefins and Alkynes: From Oxyalkynylation to Tethered Dynamic Kinetic Asymmetric Transformations (DYKAT)
Stefano Nicolai, Ugo Orcel, Bastian Muriel, Phillip D. G. Greenwood, Luca Buzzetti, Mikus Purins and Jerome Waser
Synlett 2020, in press. (DOI: 10.1055/a-1308-0021 )

Vinylbenziodoxol(on)es: Synthetic Methods and Applications
Nina Declas, Guillaume Pisella and Jerome Waser
Helv. Chim. Acta 2020, 103, e2000191. (DOI: 10.1002/hlca.202000191 )

Catalytic Enantioselective Ring-Opening Reactions of Cyclopropanes
Vincent Pirenne, Bastian Muriel, and Jerome Waser
Chem. Rev. 2020, in press. (DOI: 10.1021/acs.chemrev.0c00109 ) Green Access

Photocatalysis with organic dyes: facile access to reactive intermediates for synthesis
Stephanie G. E. Amos, Marion Garreau, Luca Buzzetti and Jerome Waser
Beilstein J. Org. Chem. 2020, 16, 1163-1187. (DOI: 10.3762/bjoc.16.103 ) Open Access!

1‐Azido‐3,3‐dimethyl‐3‐(1H )‐1,2‐benziodoxole
Raphael Simonet-Davin and Jerome Waser
Electronic Encyclopedia of Reagents for Organic Synthesis, John Wiley & Sons, 2020. (DOI: 10.1002/047084289X.rn02312 )

Publications prior to 2020

Publications 2017-2019
Publications 2013-2016
Publications 2009-2012